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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sphingosine kinase 1 (Homo sapiens (Human)) | BDBM50331854 (CHEMBL1241832 | N'-((2-hydroxynaphthalen-1-yl)meth...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet  | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.06E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pennsylvania State University College of Medicine Curated by ChEMBL | Assay Description Competitive inhibition of recombinant sphingosine kinase 1 using D-erythro-sphingosine as substrate by Lineweaver-Burk plot analysis | Bioorg Med Chem Lett 20: 7498-502 (2010) Article DOI: 10.1016/j.bmcl.2010.10.005 BindingDB Entry DOI: 10.7270/Q2J67H66 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Sphingosine kinase 1 (Homo sapiens (Human)) | BDBM50331855 (CHEMBL1289102 | N'-(1-(3,4-dimethoxyphenyl)ethylid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pennsylvania State University College of Medicine Curated by ChEMBL | Assay Description Competitive inhibition of recombinant sphingosine kinase 1 using D-erythro-sphingosine as substrate by Lineweaver-Burk plot analysis | Bioorg Med Chem Lett 20: 7498-502 (2010) Article DOI: 10.1016/j.bmcl.2010.10.005 BindingDB Entry DOI: 10.7270/Q2J67H66 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
