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PubMed code 21216504

Compile data set for download or QSAR
Found 19 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Mu-type opioid receptor


(Homo sapiens (Human))
BDBM50378890
PNG
(CHEMBL1743604)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:32,38,44,TLB:48:47:37:39.40.43|
Show InChI InChI=1S/C40H47N3O6/c1-22-16-27(44)17-23(2)28(22)20-31(41(3)4)38(46)43-21-26-9-7-6-8-24(26)18-32(43)39(47)48-34-13-10-25-19-30-29-11-12-33(45)37-40(29,14-15-42(30)5)35(25)36(34)49-37/h6-13,16-17,25,29-33,35,37,44-45H,14-15,18-21H2,1-5H3/t25?,29-,30+,31-,32-,33-,35?,37-,40-/m0/s1
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1.10n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Homo sapiens (Human))
BDBM50378889
PNG
(CHEMBL1743605)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCC(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:37,43,49,TLB:53:52:42:44.45.48|
Show InChI InChI=1S/C43H52N4O7/c1-24-18-29(48)19-25(2)30(24)22-34(45(3)4)42(52)47-23-28-9-7-6-8-26(28)20-33(47)41(51)44-16-14-37(50)53-36-13-10-27-21-32-31-11-12-35(49)40-43(31,15-17-46(32)5)38(27)39(36)54-40/h6-13,18-19,27,31-35,38,40,48-49H,14-17,20-23H2,1-5H3,(H,44,51)/t27?,31-,32+,33-,34-,35-,38?,40-,43-/m0/s1
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1.40n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO cells after 60 mins by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Homo sapiens (Human))
BDBM50378889
PNG
(CHEMBL1743605)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCC(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:37,43,49,TLB:53:52:42:44.45.48|
Show InChI InChI=1S/C43H52N4O7/c1-24-18-29(48)19-25(2)30(24)22-34(45(3)4)42(52)47-23-28-9-7-6-8-26(28)20-33(47)41(51)44-16-14-37(50)53-36-13-10-27-21-32-31-11-12-35(49)40-43(31,15-17-46(32)5)38(27)39(36)54-40/h6-13,18-19,27,31-35,38,40,48-49H,14-17,20-23H2,1-5H3,(H,44,51)/t27?,31-,32+,33-,34-,35-,38?,40-,43-/m0/s1
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1.40n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Homo sapiens (Human))
BDBM50378890
PNG
(CHEMBL1743604)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:32,38,44,TLB:48:47:37:39.40.43|
Show InChI InChI=1S/C40H47N3O6/c1-22-16-27(44)17-23(2)28(22)20-31(41(3)4)38(46)43-21-26-9-7-6-8-24(26)18-32(43)39(47)48-34-13-10-25-19-30-29-11-12-33(45)37-40(29,14-15-42(30)5)35(25)36(34)49-37/h6-13,16-17,25,29-33,35,37,44-45H,14-15,18-21H2,1-5H3/t25?,29-,30+,31-,32-,33-,35?,37-,40-/m0/s1
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1.60n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Homo sapiens (Human))
BDBM50324028
PNG
((S)-2-((S)-2-(dimethylamino)-3-(4-hydroxy-2,6-dime...)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(O)=O |r|
Show InChI InChI=1S/C23H28N2O4/c1-14-9-18(26)10-15(2)19(14)12-20(24(3)4)22(27)25-13-17-8-6-5-7-16(17)11-21(25)23(28)29/h5-10,20-21,26H,11-13H2,1-4H3,(H,28,29)/t20-,21-/m0/s1
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2.70n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(Homo sapiens (Human))
BDBM50378889
PNG
(CHEMBL1743605)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCC(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:37,43,49,TLB:53:52:42:44.45.48|
Show InChI InChI=1S/C43H52N4O7/c1-24-18-29(48)19-25(2)30(24)22-34(45(3)4)42(52)47-23-28-9-7-6-8-26(28)20-33(47)41(51)44-16-14-37(50)53-36-13-10-27-21-32-31-11-12-35(49)40-43(31,15-17-46(32)5)38(27)39(36)54-40/h6-13,18-19,27,31-35,38,40,48-49H,14-17,20-23H2,1-5H3,(H,44,51)/t27?,31-,32+,33-,34-,35-,38?,40-,43-/m0/s1
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3.5n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Homo sapiens (Human))
BDBM50378888
PNG
(CHEMBL1743603)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCC(O)=O |r|
Show InChI InChI=1S/C26H33N3O5/c1-16-11-20(30)12-17(2)21(16)14-23(28(3)4)26(34)29-15-19-8-6-5-7-18(19)13-22(29)25(33)27-10-9-24(31)32/h5-8,11-12,22-23,30H,9-10,13-15H2,1-4H3,(H,27,33)(H,31,32)/t22-,23-/m0/s1
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5.70n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Homo sapiens (Human))
BDBM50378890
PNG
(CHEMBL1743604)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:32,38,44,TLB:48:47:37:39.40.43|
Show InChI InChI=1S/C40H47N3O6/c1-22-16-27(44)17-23(2)28(22)20-31(41(3)4)38(46)43-21-26-9-7-6-8-24(26)18-32(43)39(47)48-34-13-10-25-19-30-29-11-12-33(45)37-40(29,14-15-42(30)5)35(25)36(34)49-37/h6-13,16-17,25,29-33,35,37,44-45H,14-15,18-21H2,1-5H3/t25?,29-,30+,31-,32-,33-,35?,37-,40-/m0/s1
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12n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO cells after 60 mins by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(Homo sapiens (Human))
BDBM50324028
PNG
((S)-2-((S)-2-(dimethylamino)-3-(4-hydroxy-2,6-dime...)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(O)=O |r|
Show InChI InChI=1S/C23H28N2O4/c1-14-9-18(26)10-15(2)19(14)12-20(24(3)4)22(27)25-13-17-8-6-5-7-16(17)11-21(25)23(28)29/h5-10,20-21,26H,11-13H2,1-4H3,(H,28,29)/t20-,21-/m0/s1
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2.30E+3n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(Homo sapiens (Human))
BDBM50378888
PNG
(CHEMBL1743603)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCC(O)=O |r|
Show InChI InChI=1S/C26H33N3O5/c1-16-11-20(30)12-17(2)21(16)14-23(28(3)4)26(34)29-15-19-8-6-5-7-18(19)13-22(29)25(33)27-10-9-24(31)32/h5-8,11-12,22-23,30H,9-10,13-15H2,1-4H3,(H,27,33)(H,31,32)/t22-,23-/m0/s1
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4.50E+3n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Homo sapiens (Human))
BDBM50324028
PNG
((S)-2-((S)-2-(dimethylamino)-3-(4-hydroxy-2,6-dime...)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(O)=O |r|
Show InChI InChI=1S/C23H28N2O4/c1-14-9-18(26)10-15(2)19(14)12-20(24(3)4)22(27)25-13-17-8-6-5-7-16(17)11-21(25)23(28)29/h5-10,20-21,26H,11-13H2,1-4H3,(H,28,29)/t20-,21-/m0/s1
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>1.00E+4n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO cells after 60 mins by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Homo sapiens (Human))
BDBM50378888
PNG
(CHEMBL1743603)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCC(O)=O |r|
Show InChI InChI=1S/C26H33N3O5/c1-16-11-20(30)12-17(2)21(16)14-23(28(3)4)26(34)29-15-19-8-6-5-7-18(19)13-22(29)25(33)27-10-9-24(31)32/h5-8,11-12,22-23,30H,9-10,13-15H2,1-4H3,(H,27,33)(H,31,32)/t22-,23-/m0/s1
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>1.00E+4n/an/an/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO cells after 60 mins by scintillation counting


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Homo sapiens (Human))
BDBM50378889
PNG
(CHEMBL1743605)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCC(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:37,43,49,TLB:53:52:42:44.45.48|
Show InChI InChI=1S/C43H52N4O7/c1-24-18-29(48)19-25(2)30(24)22-34(45(3)4)42(52)47-23-28-9-7-6-8-26(28)20-33(47)41(51)44-16-14-37(50)53-36-13-10-27-21-32-31-11-12-35(49)40-43(31,15-17-46(32)5)38(27)39(36)54-40/h6-13,18-19,27,31-35,38,40,48-49H,14-17,20-23H2,1-5H3,(H,44,51)/t27?,31-,32+,33-,34-,35-,38?,40-,43-/m0/s1
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n/an/a 0.810n/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Antagonist activity at human delta opioid receptor expressed in CHO cells assessed as inhibition of U50488-induced [35S]GTPgammaS binding


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Homo sapiens (Human))
BDBM50378890
PNG
(CHEMBL1743604)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:32,38,44,TLB:48:47:37:39.40.43|
Show InChI InChI=1S/C40H47N3O6/c1-22-16-27(44)17-23(2)28(22)20-31(41(3)4)38(46)43-21-26-9-7-6-8-24(26)18-32(43)39(47)48-34-13-10-25-19-30-29-11-12-33(45)37-40(29,14-15-42(30)5)35(25)36(34)49-37/h6-13,16-17,25,29-33,35,37,44-45H,14-15,18-21H2,1-5H3/t25?,29-,30+,31-,32-,33-,35?,37-,40-/m0/s1
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n/an/a 1.70n/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Antagonist activity at human delta opioid receptor expressed in CHO cells assessed as inhibition of U50488-induced [35S]GTPgammaS binding


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(Homo sapiens (Human))
BDBM50378890
PNG
(CHEMBL1743604)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:32,38,44,TLB:48:47:37:39.40.43|
Show InChI InChI=1S/C40H47N3O6/c1-22-16-27(44)17-23(2)28(22)20-31(41(3)4)38(46)43-21-26-9-7-6-8-24(26)18-32(43)39(47)48-34-13-10-25-19-30-29-11-12-33(45)37-40(29,14-15-42(30)5)35(25)36(34)49-37/h6-13,16-17,25,29-33,35,37,44-45H,14-15,18-21H2,1-5H3/t25?,29-,30+,31-,32-,33-,35?,37-,40-/m0/s1
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n/an/a 13n/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Agonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assay


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(Homo sapiens (Human))
BDBM50378889
PNG
(CHEMBL1743605)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCC(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:37,43,49,TLB:53:52:42:44.45.48|
Show InChI InChI=1S/C43H52N4O7/c1-24-18-29(48)19-25(2)30(24)22-34(45(3)4)42(52)47-23-28-9-7-6-8-26(28)20-33(47)41(51)44-16-14-37(50)53-36-13-10-27-21-32-31-11-12-35(49)40-43(31,15-17-46(32)5)38(27)39(36)54-40/h6-13,18-19,27,31-35,38,40,48-49H,14-17,20-23H2,1-5H3,(H,44,51)/t27?,31-,32+,33-,34-,35-,38?,40-,43-/m0/s1
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n/an/a 450n/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Agonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assay


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Homo sapiens (Human))
BDBM50378890
PNG
(CHEMBL1743604)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:32,38,44,TLB:48:47:37:39.40.43|
Show InChI InChI=1S/C40H47N3O6/c1-22-16-27(44)17-23(2)28(22)20-31(41(3)4)38(46)43-21-26-9-7-6-8-24(26)18-32(43)39(47)48-34-13-10-25-19-30-29-11-12-33(45)37-40(29,14-15-42(30)5)35(25)36(34)49-37/h6-13,16-17,25,29-33,35,37,44-45H,14-15,18-21H2,1-5H3/t25?,29-,30+,31-,32-,33-,35?,37-,40-/m0/s1
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n/an/a 3.10E+3n/an/an/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Antagonist activity at human kappa opioid receptor expressed in CHO cells assessed as inhibition of SNC80-induced [35S]GTPgammaS binding


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Homo sapiens (Human))
BDBM50378889
PNG
(CHEMBL1743605)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCC(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:37,43,49,TLB:53:52:42:44.45.48|
Show InChI InChI=1S/C43H52N4O7/c1-24-18-29(48)19-25(2)30(24)22-34(45(3)4)42(52)47-23-28-9-7-6-8-26(28)20-33(47)41(51)44-16-14-37(50)53-36-13-10-27-21-32-31-11-12-35(49)40-43(31,15-17-46(32)5)38(27)39(36)54-40/h6-13,18-19,27,31-35,38,40,48-49H,14-17,20-23H2,1-5H3,(H,44,51)/t27?,31-,32+,33-,34-,35-,38?,40-,43-/m0/s1
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n/an/an/an/a 20n/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Agonist activity at human kappa opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assay


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(Homo sapiens (Human))
BDBM50378889
PNG
(CHEMBL1743605)
Show SMILES CN(C)[C@@H](Cc1c(C)cc(O)cc1C)C(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCC(=O)OC1=C2O[C@H]3[C@@H](O)C=C[C@H]4[C@H]5CC(C=C1)C2[C@@]34CCN5C |r,c:37,43,49,TLB:53:52:42:44.45.48|
Show InChI InChI=1S/C43H52N4O7/c1-24-18-29(48)19-25(2)30(24)22-34(45(3)4)42(52)47-23-28-9-7-6-8-26(28)20-33(47)41(51)44-16-14-37(50)53-36-13-10-27-21-32-31-11-12-35(49)40-43(31,15-17-46(32)5)38(27)39(36)54-40/h6-13,18-19,27,31-35,38,40,48-49H,14-17,20-23H2,1-5H3,(H,44,51)/t27?,31-,32+,33-,34-,35-,38?,40-,43-/m0/s1
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UniProtKB/SwissProt

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n/an/an/an/a 29n/an/an/an/a



University of Cagliari

Curated by ChEMBL


Assay Description
Agonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assay


Eur J Med Chem 46: 799-803 (2011)


Article DOI: 10.1016/j.ejmech.2010.12.001
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%