Found 20 hits of Enzyme Inhibition Constant Data Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339279
(5-(Chloromethyl)-3-(naphthalen-1-yl)-2-(trifluorom...)Show SMILES FC(F)(F)c1[nH]n2c(nc(CCl)cc2=O)c1-c1cccc2ccccc12 |(-2.75,-35.11,;-3.52,-36.45,;-5.06,-36.46,;-4.3,-35.1,;-2.74,-37.78,;-3.35,-39.19,;-2.2,-40.22,;-.88,-39.44,;.46,-40.22,;.46,-41.77,;1.8,-42.54,;3.14,-41.77,;-.88,-42.53,;-2.21,-41.77,;-3.55,-42.54,;-1.2,-37.94,;-.37,-36.63,;-1.09,-35.27,;-.27,-33.97,;1.29,-34.03,;2,-35.4,;3.53,-35.47,;4.24,-36.83,;3.42,-38.13,;1.88,-38.06,;1.17,-36.7,)| Show InChI InChI=1S/C18H11ClF3N3O/c19-9-11-8-14(26)25-17(23-11)15(16(24-25)18(20,21)22)13-7-3-5-10-4-1-2-6-12(10)13/h1-8,24H,9H2 | PDB
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PubMed
| n/a | n/a | n/a | n/a | 1.25E+3 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 1
(Homo sapiens (Human)) | BDBM50339281
(5-(2,6-Dichloro-5-fluoropyridin-3-yl)-3-phenyl-2-(...)Show SMILES Fc1cc(c(Cl)nc1Cl)-c1cc(=O)n2[nH]c(c(-c3ccccc3)c2n1)C(F)(F)F Show InChI InChI=1S/C18H8Cl2F4N4O/c19-15-9(6-10(21)16(20)26-15)11-7-12(29)28-17(25-11)13(8-4-2-1-3-5-8)14(27-28)18(22,23)24/h1-7,27H | PDB
Reactome pathway
KEGG
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| n/a | n/a | n/a | n/a | 4.93E+4 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ1 expressed in HEK293 cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339277
(5-(Chloromethyl)-3-phenyl-2-(trifluoromethyl)pyraz...)Show InChI InChI=1S/C14H9ClF3N3O/c15-7-9-6-10(22)21-13(19-9)11(8-4-2-1-3-5-8)12(20-21)14(16,17)18/h1-6,20H,7H2 | PDB
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| n/a | n/a | n/a | n/a | 2.27E+3 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339283
(5-(chloromethyl)-3-(4-chlorophenyl)-2-(trifluorome...)Show SMILES FC(F)(F)c1[nH]n2c(nc(CCl)cc2=O)c1-c1ccc(Cl)cc1 Show InChI InChI=1S/C14H8Cl2F3N3O/c15-6-9-5-10(23)22-13(20-9)11(12(21-22)14(17,18)19)7-1-3-8(16)4-2-7/h1-5,21H,6H2 | PDB
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| n/a | n/a | n/a | n/a | 2.33E+3 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339293
(3-(4-Chlorophenyl)-2,5-bis(trifluoromethyl)pyrazol...)Show SMILES FC(F)(F)c1[nH]n2c(nc(cc2=O)C(F)(F)F)c1-c1ccc(Cl)cc1 Show InChI InChI=1S/C14H6ClF6N3O/c15-7-3-1-6(2-4-7)10-11(14(19,20)21)23-24-9(25)5-8(13(16,17)18)22-12(10)24/h1-5,23H | PDB
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| n/a | n/a | n/a | n/a | 2.06E+3 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339281
(5-(2,6-Dichloro-5-fluoropyridin-3-yl)-3-phenyl-2-(...)Show SMILES Fc1cc(c(Cl)nc1Cl)-c1cc(=O)n2[nH]c(c(-c3ccccc3)c2n1)C(F)(F)F Show InChI InChI=1S/C18H8Cl2F4N4O/c19-15-9(6-10(21)16(20)26-15)11-7-12(29)28-17(25-11)13(8-4-2-1-3-5-8)14(27-28)18(22,23)24/h1-7,27H | PDB
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| n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339285
(5-tert-Butyl-3-phenyl-2-(trifluoromethyl)pyrazolo[...)Show SMILES CC(C)(C)c1cc(=O)n2[nH]c(c(-c3ccccc3)c2n1)C(F)(F)F Show InChI InChI=1S/C17H16F3N3O/c1-16(2,3)11-9-12(24)23-15(21-11)13(10-7-5-4-6-8-10)14(22-23)17(18,19)20/h4-9,22H,1-3H3 | PDB
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| n/a | n/a | n/a | n/a | 6.19E+3 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339286
(5-(Difluoromethyl)-3-phenyl-2-(trifluoromethyl)pyr...)Show SMILES FC(F)c1cc(=O)n2[nH]c(c(-c3ccccc3)c2n1)C(F)(F)F Show InChI InChI=1S/C14H8F5N3O/c15-12(16)8-6-9(23)22-13(20-8)10(7-4-2-1-3-5-7)11(21-22)14(17,18)19/h1-6,12,21H | PDB
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| n/a | n/a | n/a | n/a | 4.29E+3 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339291
(5-(2,3,4,5-Tetrafluorophenyl)-3-(thiophen-2-yl)-2-...)Show SMILES Fc1cc(c(F)c(F)c1F)-c1cc(=O)n2[nH]c(c(-c3cccs3)c2n1)C(F)(F)F Show InChI InChI=1S/C17H6F7N3OS/c18-7-4-6(12(19)14(21)13(7)20)8-5-10(28)27-16(25-8)11(9-2-1-3-29-9)15(26-27)17(22,23)24/h1-5,26H | PDB
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| n/a | n/a | n/a | n/a | 160 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339292
(5-tert-Butyl-3-(naphthalen-1-yl)-2-(trifluoromethy...)Show SMILES CC(C)(C)c1cc(=O)n2[nH]c(c(-c3cccc4ccccc34)c2n1)C(F)(F)F |(31.87,-46.88,;31.87,-45.34,;33.21,-44.57,;33.2,-46.11,;30.53,-44.56,;29.2,-45.33,;27.86,-44.56,;26.53,-45.34,;27.87,-43.01,;26.72,-41.99,;27.34,-40.58,;28.87,-40.74,;29.79,-39.5,;29.17,-38.09,;30.09,-36.85,;31.63,-37.02,;32.24,-38.44,;33.77,-38.62,;34.38,-40.03,;33.45,-41.27,;31.92,-41.08,;31.32,-39.67,;29.2,-42.24,;30.53,-43.02,;26.56,-39.25,;27.32,-37.91,;25.02,-39.26,;25.77,-37.91,)| Show InChI InChI=1S/C21H18F3N3O/c1-20(2,3)15-11-16(28)27-19(25-15)17(18(26-27)21(22,23)24)14-10-6-8-12-7-4-5-9-13(12)14/h4-11,26H,1-3H3 | PDB
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| n/a | n/a | n/a | n/a | 1.93E+4 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339282
(5-(2,6-Dichloro-5-fluoropyridin-3-yl)-3-(naphthale...)Show SMILES Fc1cc(c(Cl)nc1Cl)-c1cc(=O)n2[nH]c(c(-c3cccc4ccccc34)c2n1)C(F)(F)F |(3.56,-4.78,;2.23,-5.55,;.89,-4.79,;-.44,-5.56,;-.44,-7.1,;-1.78,-7.87,;.89,-7.88,;2.23,-7.11,;3.57,-7.88,;-1.77,-4.79,;-3.1,-5.55,;-4.43,-4.79,;-5.77,-5.56,;-4.43,-3.24,;-5.57,-2.22,;-4.96,-.81,;-3.43,-.96,;-2.6,.34,;-3.32,1.7,;-2.5,3,;-.95,2.93,;-.23,1.57,;1.3,1.51,;2.01,.15,;1.19,-1.16,;-.35,-1.09,;-1.06,.27,;-3.1,-2.46,;-1.77,-3.24,;-5.74,.52,;-4.97,1.86,;-7.28,.51,;-6.52,1.86,)| Show InChI InChI=1S/C22H10Cl2F4N4O/c23-19-13(8-14(25)20(24)30-19)15-9-16(33)32-21(29-15)17(18(31-32)22(26,27)28)12-7-3-5-10-4-1-2-6-11(10)12/h1-9,31H | PDB
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| n/a | n/a | n/a | n/a | 150 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339289
(5-(2,6-Dichloro-5-fluoropyridin-3-yl)-3-(3,4-dimet...)Show SMILES COc1ccc(cc1OC)-c1c([nH]n2c1nc(cc2=O)-c1cc(F)c(Cl)nc1Cl)C(F)(F)F Show InChI InChI=1S/C20H12Cl2F4N4O3/c1-32-12-4-3-8(5-13(12)33-2)15-16(20(24,25)26)29-30-14(31)7-11(27-19(15)30)9-6-10(23)18(22)28-17(9)21/h3-7,29H,1-2H3 | PDB
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| n/a | n/a | n/a | n/a | 230 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339280
(3-(Naphthalen-1-yl)-2,5-bis(trifluoromethyl)pyrazo...)Show SMILES FC(F)(F)c1[nH]n2c(nc(cc2=O)C(F)(F)F)c1-c1cccc2ccccc12 |(12.13,-33.97,;11.37,-35.32,;9.82,-35.33,;10.58,-33.97,;12.15,-36.65,;11.53,-38.06,;12.68,-39.08,;14.01,-38.31,;15.34,-39.09,;15.34,-40.63,;14.01,-41.4,;12.67,-40.63,;11.33,-41.41,;16.68,-41.41,;16.68,-42.96,;18.02,-40.64,;18.02,-42.18,;13.68,-36.8,;14.51,-35.5,;13.79,-34.14,;14.62,-32.83,;16.17,-32.9,;16.88,-34.27,;18.41,-34.34,;19.13,-35.69,;18.3,-37,;16.76,-36.93,;16.05,-35.57,)| Show InChI InChI=1S/C18H9F6N3O/c19-17(20,21)12-8-13(28)27-16(25-12)14(15(26-27)18(22,23)24)11-7-3-5-9-4-1-2-6-10(9)11/h1-8,26H | PDB
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| n/a | n/a | n/a | n/a | 4.98E+3 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50143558
(CHEMBL41355 | EZOGABINE | N-(2-amino-4-(4-fluorobe...)Show InChI InChI=1S/C16H18FN3O2/c1-2-22-16(21)20-15-8-7-13(9-14(15)18)19-10-11-3-5-12(17)6-4-11/h3-9,19H,2,10,18H2,1H3,(H,20,21) | PDB
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| n/a | n/a | n/a | n/a | 430 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | 
3D Structure (crystal) |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339290
(5-(3-Nitrophenyl)-3-(thiophen-2-yl)-2-(trifluorome...)Show SMILES [O-][N+](=O)c1cccc(c1)-c1cc(=O)n2[nH]c(c(-c3cccs3)c2n1)C(F)(F)F Show InChI InChI=1S/C17H9F3N4O3S/c18-17(19,20)15-14(12-5-2-6-28-12)16-21-11(8-13(25)23(16)22-15)9-3-1-4-10(7-9)24(26)27/h1-8,22H | PDB
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| n/a | n/a | n/a | n/a | 580 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339294
(3-(4-Chlorophenyl)-2-(trifluoromethyl)-5-(2,4,5-tr...)Show SMILES Fc1cc(F)c(cc1F)-c1cc(=O)n2[nH]c(c(-c3ccc(Cl)cc3)c2n1)C(F)(F)F Show InChI InChI=1S/C19H8ClF6N3O/c20-9-3-1-8(2-4-9)16-17(19(24,25)26)28-29-15(30)7-14(27-18(16)29)10-5-12(22)13(23)6-11(10)21/h1-7,28H | PDB
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| n/a | n/a | n/a | n/a | 210 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339278
(3-Phenyl-2,5-bis(trifluoromethyl)pyrazolo[1,5-a]py...)Show SMILES FC(F)(F)c1[nH]n2c(nc(cc2=O)C(F)(F)F)c1-c1ccccc1 Show InChI InChI=1S/C14H7F6N3O/c15-13(16,17)8-6-9(24)23-12(21-8)10(7-4-2-1-3-5-7)11(22-23)14(18,19)20/h1-6,22H | PDB
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CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | n/a | n/a | 1.46E+3 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339284
(5-(4-Methoxyphenyl)-3-phenyl-2-(trifluoromethyl)py...)Show SMILES COc1ccc(cc1)-c1cc(=O)n2[nH]c(c(-c3ccccc3)c2n1)C(F)(F)F Show InChI InChI=1S/C20H14F3N3O2/c1-28-14-9-7-12(8-10-14)15-11-16(27)26-19(24-15)17(13-5-3-2-4-6-13)18(25-26)20(21,22)23/h2-11,25H,1H3 | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | n/a | n/a | 1.93E+3 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339288
(5-(3-Nitrophenyl)-3-phenyl-2-(trifluoromethyl)pyra...)Show SMILES [O-][N+](=O)c1cccc(c1)-c1cc(=O)n2[nH]c(c(-c3ccccc3)c2n1)C(F)(F)F Show InChI InChI=1S/C19H11F3N4O3/c20-19(21,22)17-16(11-5-2-1-3-6-11)18-23-14(10-15(27)25(18)24-17)12-7-4-8-13(9-12)26(28)29/h1-10,24H | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | n/a | n/a | 570 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily KQT member 2/3
(Homo sapiens (Human)) | BDBM50339287
(3-Phenyl-5-(2,3,4,5-tetrafluorophenyl)-2-(trifluor...)Show SMILES Fc1cc(-c2cc(=O)n3[nH]c(c(-c4ccccc4)c3n2)C(F)(F)F)c(F)c(F)c1F Show InChI InChI=1S/C19H8F7N3O/c20-10-6-9(14(21)16(23)15(10)22)11-7-12(30)29-18(27-11)13(8-4-2-1-3-5-8)17(28-29)19(24,25)26/h1-7,28H | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | n/a | n/a | 600 | n/a | n/a | n/a | n/a |
Hebei Medical University
Curated by ChEMBL
| Assay Description
Activation of KCNQ2/Q3 expressed in CHO cells by atomic absorption Rb'+ efflux assay |
Eur J Med Chem 46: 934-43 (2011)
Article DOI: 10.1016/j.ejmech.2011.01.010
BindingDB Entry DOI: 10.7270/Q2TM7BDF |
More data for this
Ligand-Target Pair | |
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