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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Vascular endothelial growth factor receptor 2 (Homo sapiens (Human)) | BDBM50338503 (4-(pyridin-4-ylmethylthio)-N-(3-(trifluoromethyl)p...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet  | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 309 | n/a | n/a | n/a | n/a | n/a | n/a |
Santen Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of KDR assessed as phosphorylation level of substrate by ELISA | Bioorg Med Chem Lett 21: 1782-5 (2011) Article DOI: 10.1016/j.bmcl.2011.01.063 BindingDB Entry DOI: 10.7270/Q2DN45BZ | |||||||||||
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