Affinity Data by PubMed id=21530277

PubMed code 21530277

Found 3 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Multidrug resistance-associated protein 1 (Homo sapiens (Human))	BDBM50349861 (CHEMBL1813579) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	660	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kakatiya University Curated by ChEMBL					Assay Description Inhibition of human MRP1 expressed in Spodoptera frugiperda Sf9 cells assessed as inhibition of NEM-GS-induced vanadate-sensitive ATPase activity mea...				Bioorg Med Chem 19: 3249-54 (2011) Article DOI: 10.1016/j.bmc.2011.03.051 BindingDB Entry DOI: 10.7270/Q29P3208
Kakatiya University Curated by ChEMBL					More data for this Ligand-Target Pair
Multidrug resistance-associated protein 1 (Homo sapiens (Human))	BDBM50349860 (CHEMBL1770422) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	950	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kakatiya University Curated by ChEMBL					Assay Description Inhibition of human MRP1 expressed in Spodoptera frugiperda Sf9 cells assessed as inhibition of NEM-GS-induced vanadate-sensitive ATPase activity mea...				Bioorg Med Chem 19: 3249-54 (2011) Article DOI: 10.1016/j.bmc.2011.03.051 BindingDB Entry DOI: 10.7270/Q29P3208
Kakatiya University Curated by ChEMBL					More data for this Ligand-Target Pair
Multidrug resistance-associated protein 1 (Homo sapiens (Human))	BDBM50158460 ((3,5-dibromo-4-hydroxyphenyl)(2-ethyl-1-benzofuran...) Show SMILES CCc1oc2ccccc2c1C(=O)c1cc(Br)c(O)c(Br)c1 Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	4.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Kakatiya University Curated by ChEMBL					Assay Description Inhibition of human MRP1 expressed in Spodoptera frugiperda Sf9 cells assessed as inhibition of NEM-GS-induced vanadate-sensitive ATPase activity mea...				Bioorg Med Chem 19: 3249-54 (2011) Article DOI: 10.1016/j.bmc.2011.03.051 BindingDB Entry DOI: 10.7270/Q29P3208
Kakatiya University Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%