Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
cAMP-dependent protein kinase catalytic subunit alpha (Homo sapiens (Human)) | BDBM15211 (CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank MMDB PDB PubMed | 48 | -42.5 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
cAMP-dependent protein kinase catalytic subunit alpha (Homo sapiens (Human)) | BDBM92607 (H-88) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | 360 | -37.4 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase 1 (Homo sapiens (Human)) | BDBM15211 (CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 480 | -36.7 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase 1 (Homo sapiens (Human)) | BDBM92607 (H-88) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | 760 | -35.5 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myosin light chain kinase 3 (Homo sapiens (Human)) | BDBM15211 (CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 2.83E+4 | -26.4 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcium/calmodulin-dependent protein kinase type II subunit beta (Homo sapiens (Human)) | BDBM15211 (CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 2.97E+4 | -26.3 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Homo sapiens (Human)) | BDBM15211 (CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 3.17E+4 | -26.1 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase I isoform alpha (Homo sapiens (Human)) | BDBM15211 (CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 3.83E+4 | -25.6 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myosin light chain kinase 3 (Homo sapiens (Human)) | BDBM92607 (H-88) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | 5.00E+4 | -25.0 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase I isoform alpha (Homo sapiens (Human)) | BDBM92607 (H-88) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | 6.07E+4 | -24.5 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcium/calmodulin-dependent protein kinase type II subunit beta (Homo sapiens (Human)) | BDBM92607 (H-88) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | 7.13E+4 | -24.1 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Homo sapiens (Human)) | BDBM92607 (H-88) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | 7.57E+4 | -23.9 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha (Homo sapiens (Human)) | BDBM92607 (H-88) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | 1.04E+5 | -23.1 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha (Homo sapiens (Human)) | BDBM15211 (CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 1.37E+5 | -22.4 | n/a | n/a | n/a | n/a | n/a | n/a | 30 |
Nagoya University School of Medicine | Assay Description Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d... | J Biol Chem 265: 5267-72 (1990) BindingDB Entry DOI: 10.7270/Q2QR4VRF | |||||||||||
More data for this Ligand-Target Pair |