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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50349897 (CHEMBL1814705) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet  | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50000092 ((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB Article PubMed | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair |  3D Structure (crystal) | ||||||||||||
| Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50349897 (CHEMBL1814705) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 51 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50349896 (CHEMBL1814704) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 67 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50349894 (CHEMBL1814702) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 619 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50349895 (CHEMBL1814703) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.08E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50349896 (CHEMBL1814704) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50349897 (CHEMBL1814705) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in recombinant hDOR-CHO cells after 2 hrs by liquid scintillation co... | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50349896 (CHEMBL1814704) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in recombinant hDOR-CHO cells after 2 hrs by liquid scintillation co... | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50349895 (CHEMBL1814703) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50349894 (CHEMBL1814702) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in recombinant hDOR-CHO cells after 2 hrs by liquid scintillation co... | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50349895 (CHEMBL1814703) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in recombinant hDOR-CHO cells after 2 hrs by liquid scintillation co... | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50349894 (CHEMBL1814702) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute on Drug Abuse and The National Institute on Alcohol Abuse and Alcoholism Curated by ChEMBL | Assay Description Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting | Bioorg Med Chem 19: 3434-43 (2011) Article DOI: 10.1016/j.bmc.2011.04.028 BindingDB Entry DOI: 10.7270/Q2SQ90SQ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
