Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Kinesin-like protein KIF11 (Homo sapiens (Human)) | BDBM50361463 (CHEMBL1938593) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Medical University of Silesia Curated by ChEMBL | Assay Description Inhibition of mitotic kinesin Eg5 in human transformed WI38VA13 cells assessed as inhibition of microtubule-activated ATPase activity | Eur J Med Chem 46: 3179-89 (2011) Article DOI: 10.1016/j.ejmech.2011.05.013 BindingDB Entry DOI: 10.7270/Q2SB465F | |||||||||||
More data for this Ligand-Target Pair |