Affinity Data by PubMed id=21664823

PubMed code 21664823

Found 15 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347195 (CHEMBL1795747) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	96	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347200 (CHEMBL1795752) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	190	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50098126 (2-(morpholin-4-yl)-benzo[h]chromen-4-one \| 2-Morph...) Show SMILES O=c1cc(oc2c3ccccc3ccc12)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	300	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of DNA-PK				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347198 (CHEMBL1795750) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	330	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50159668 (2-Morpholin-4-yl-benzo[g]chromen-4-one \| 2-morphol...) Show SMILES O=c1cc(oc2cc3ccccc3cc12)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	400	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of DNA-PK				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347191 (CHEMBL1795743) Show SMILES O=c1nc(oc2c3ccccc3ccc12)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	420	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347194 (CHEMBL1795746) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	717	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347190 (CHEMBL1795742) Show SMILES O=c1nc(oc2ccc3ccccc3c12)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	720	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347199 (CHEMBL1795751) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	760	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347197 (CHEMBL1795749) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	930	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347196 (CHEMBL1795748) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.70E+3	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347193 (CHEMBL1795745) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.43E+3	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347201 (CHEMBL1795753) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.09E+3	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50159678 (3-Morpholin-4-yl-benzo[f]chromen-1-one \| 3-morphol...) Show SMILES O=c1cc(oc2ccc3ccccc3c12)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	4.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of DNA-PK				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair
DNA-dependent protein kinase catalytic subunit (Homo sapiens (Human))	BDBM50347192 (CHEMBL1795744) Show SMILES O=c1nc(oc2cc3ccccc3cc12)N1CCOCC1 Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
La Trobe University Curated by ChEMBL					Assay Description Inhibition of purified DNA-PK by ADP-Glo Kinase assay				Bioorg Med Chem 19: 3983-94 (2011) Article DOI: 10.1016/j.bmc.2011.05.032 BindingDB Entry DOI: 10.7270/Q20Z73M7
La Trobe University Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%