Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transcription factor Jun (Homo sapiens (Human)) | BDBM50352478 (CHEMBL1823866) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
NCI-Frederick Curated by ChEMBL | Assay Description Inhibition of AP1 expressed in HEK293T cells coexpressing beta-lactamase pre-incubated 1 hr before TPA addition measured 18 hrs post TPA challenge by... | J Nat Prod 74: 1686-91 (2011) Article DOI: 10.1021/np2005083 BindingDB Entry DOI: 10.7270/Q2GM87P2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription factor Jun (Homo sapiens (Human)) | BDBM50352479 (CHEMBL1823867) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
NCI-Frederick Curated by ChEMBL | Assay Description Inhibition of AP1 expressed in HEK293T cells coexpressing beta-lactamase pre-incubated 1 hr before TPA addition measured 18 hrs post TPA challenge by... | J Nat Prod 74: 1686-91 (2011) Article DOI: 10.1021/np2005083 BindingDB Entry DOI: 10.7270/Q2GM87P2 | |||||||||||
More data for this Ligand-Target Pair |