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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237346 (3-(4-Chlorobenzo[d]thiazol-2-yl)-2-(2-chloro-6-flu...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet  | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237348 (3-(6-Fluorobenzo[d]thiazol-2-yl)-2-(2,6-dichloroph...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM1434 (11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair |  3D Structure (crystal) | ||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237352 (3-(4-Methoxybenzo[d]thiazol-2-yl)-2-(2,6-dichlorop...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237354 (3-(6-Ethoxybenzo[d]thiazol-2-yl)-2-(2-chloro-6-flu...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.40E+3 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237344 (3-(6-Chlorobenzo[d]thiazol-2-yl)-2-(2-chloro-6-flu...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237351 (3-(6-Methoxybenzo[d]thiazol-2-yl)-2-(2,6-difluorop...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237353 (3-(4-Methoxybenzo[d]thiazol-2-yl)-2-(2-chloro-6-fl...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237347 (3-(4-Chlorobenzo[d]thiazol-2-yl)-2-(2,6-difluoroph...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237350 (3-(6-Methoxybenzo[d]thiazol-2-yl)-2-(2-chloro-6-fl...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237341 (3-(Benzo[d]thiazol-2-yl)-2-(2,6-difluorophenyl)thi...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237349 (3-(6-Methoxybenzo[d]thiazol-2-yl)-2-(2,6-dichlorop...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237342 (3-(Benzo[d]thiazol-2-yl)-2-(2-chloro-6-fluoropheny...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237345 (3-(4-Chlorobenzo[d]thiazol-2-yl)-2-(2,6-dichloroph...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237343 (3-(6-Chlorobenzo[d]thiazol-2-yl)-2-(2,6-dichloroph...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Gag-Pol polyprotein (Human immunodeficiency virus type 1 group M subtyp...) | BDBM237355 (3-(6-Ethoxybenzo[d]thiazol-2-yl)-2-(2,6-difluoroph...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | 7.8 | 37 |
Aristotle University of Thessaloniki | Assay Description HIV-1 Reverse Transcriptase Activity was measured using the colorimetric photometric immunoassay kit provided by Roche. Estimation of RT activity is ... | J Enzyme Inhib Med Chem 28: 113-22 (2013) Article DOI: 10.3109/14756366.2011.636362 BindingDB Entry DOI: 10.7270/Q2PR7TV6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
