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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Prothrombin (Homo sapiens (Human)) | BDBM50350223 (CHEMBL1812010) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet  | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University Curated by ChEMBL | Assay Description Inhibition of recombinant wild type thrombin expressed in BHK cells assessed as spectrozyme TH hydrolysis after 10 mins | J Med Chem 55: 6888-97 (2012) Article DOI: 10.1021/jm300670q BindingDB Entry DOI: 10.7270/Q2TH8NTW | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Coagulation factor X (Homo sapiens (Human)) | BDBM50350223 (CHEMBL1812010) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University Curated by ChEMBL | Assay Description Inhibition of human plasma F10a assessed as spectrozyme TH hydrolysis after 10 mins | J Med Chem 55: 6888-97 (2012) Article DOI: 10.1021/jm300670q BindingDB Entry DOI: 10.7270/Q2TH8NTW | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
