Affinity Data by PubMed id=23017884

PubMed code 23017884

Found 4 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mu-type opioid receptor (Homo sapiens (Human))	BDBM50394031 (CHEMBL2158541) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	400	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Displacement of [3H]DAMGO from human recombinant mu-opioid receptor expressed in CHO cells after 60 mins by liquid scintillation assay				Bioorg Med Chem Lett 22: 6580-2 (2012) Article DOI: 10.1016/j.bmcl.2012.09.008 BindingDB Entry DOI: 10.7270/Q2V9896X
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Homo sapiens (Human))	BDBM50394031 (CHEMBL2158541) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	>5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Displacement of [3H]DPDPE from human recombinant kappa-opioid receptor expressed in CHO cells after 60 mins by liquid scintillation assay				Bioorg Med Chem Lett 22: 6580-2 (2012) Article DOI: 10.1016/j.bmcl.2012.09.008 BindingDB Entry DOI: 10.7270/Q2V9896X
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50394031 (CHEMBL2158541) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	>5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Displacement of [3H]-U69593 from human recombinant delta-opioid receptor expressed in CHO cells after 60 mins by liquid scintillation assay				Bioorg Med Chem Lett 22: 6580-2 (2012) Article DOI: 10.1016/j.bmcl.2012.09.008 BindingDB Entry DOI: 10.7270/Q2V9896X
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (Homo sapiens (Human))	BDBM50394031 (CHEMBL2158541) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Displacement of [3H]DAMGO from human recombinant mu-opioid receptor expressed in CHO cells after 60 mins by liquid scintillation assay				Bioorg Med Chem Lett 22: 6580-2 (2012) Article DOI: 10.1016/j.bmcl.2012.09.008 BindingDB Entry DOI: 10.7270/Q2V9896X
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%