Affinity Data by PubMed id=23072958

PubMed code 23072958

Found 24 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401540 (CHEMBL2207073) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.40E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401540 (CHEMBL2207073) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.41E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401541 (CHEMBL2207074) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.62E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401541 (CHEMBL2207074) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.70E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 2 (Homo sapiens (Human))	BDBM50401541 (CHEMBL2207074) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT2 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 2 (Homo sapiens (Human))	BDBM50401543 (CHEMBL2207076) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT2 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 3 (Homo sapiens (Human))	BDBM50401543 (CHEMBL2207076) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT3 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 2 (Homo sapiens (Human))	BDBM50401544 (CHEMBL2207077) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT2 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401545 (CHEMBL2207078) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401544 (CHEMBL2207077) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 3 (Homo sapiens (Human))	BDBM50401541 (CHEMBL2207074) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT3 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 3 (Homo sapiens (Human))	BDBM50401544 (CHEMBL2207077) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT3 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 2 (Homo sapiens (Human))	BDBM50401540 (CHEMBL2207073) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT2 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 3 (Homo sapiens (Human))	BDBM50401545 (CHEMBL2207078) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT3 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401543 (CHEMBL2207076) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401542 (CHEMBL2207075) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 3 (Homo sapiens (Human))	BDBM50401540 (CHEMBL2207073) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT3 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 3 (Homo sapiens (Human))	BDBM50401542 (CHEMBL2207075) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT3 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 2 (Homo sapiens (Human))	BDBM50401542 (CHEMBL2207075) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT2 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 2 (Homo sapiens (Human))	BDBM50401545 (CHEMBL2207078) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT2 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401544 (CHEMBL2207077) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.16E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401542 (CHEMBL2207075) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.16E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401545 (CHEMBL2207078) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.16E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Homo sapiens (Human))	BDBM50401543 (CHEMBL2207076) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.16E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting				Bioorg Med Chem 20: 6831-9 (2012) Article DOI: 10.1016/j.bmc.2012.09.049 BindingDB Entry DOI: 10.7270/Q25B03PT
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%