Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432959 (CHEMBL2377726) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432963 (CHEMBL2377752) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 80 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432971 (CHEMBL2377745) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 90 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432972 (CHEMBL2377744) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432975 (CHEMBL2377741) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432955 (CHEMBL2377730) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432965 (CHEMBL2377750) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432949 (CHEMBL2377736) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432958 (CHEMBL2377727) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 80 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432961 (CHEMBL2375386) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432968 (CHEMBL2377748) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432973 (CHEMBL2377743) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432976 (CHEMBL2377740) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432978 (CHEMBL2377738) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432950 (CHEMBL2377735) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432956 (CHEMBL2377729) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 400 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432957 (CHEMBL2377728) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 450 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432970 (CHEMBL2377746) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432951 (CHEMBL2377734) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 400 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432952 (CHEMBL2377733) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432953 (CHEMBL2377732) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432954 (CHEMBL2377731) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432960 (KRN-568 | NPS-R-568 | Norcalcin | R-568 | TECALCET...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 80 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432966 (CHEMBL2375383) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432974 (CHEMBL2377742) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 600 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432948 (CHEMBL2377737) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 150 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432969 (CHEMBL2377747) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 80 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432977 (CHEMBL2377739) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 80 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432967 (CHEMBL2377749) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432962 (CHEMBL2375385) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Extracellular calcium-sensing receptor (Homo sapiens (Human)) | BDBM50432964 (CHEMBL2377751) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Galapagos SASU Curated by ChEMBL | Assay Description Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep... | Bioorg Med Chem Lett 23: 2455-9 (2013) Article DOI: 10.1016/j.bmcl.2013.01.077 BindingDB Entry DOI: 10.7270/Q228090Q | |||||||||||
More data for this Ligand-Target Pair |