Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutamate carboxypeptidase 2 (Homo sapiens (Human)) | BDBM17755 (2-(3-sulfanylpropyl)pentanedioic acid | 2-MPPA | C...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins University Curated by ChEMBL | Assay Description Inhibition of GCP2 (unknown origin) | J Med Chem 57: 243-7 (2014) Article DOI: 10.1021/jm401703a BindingDB Entry DOI: 10.7270/Q2HH6MJB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate carboxypeptidase 2 (Homo sapiens (Human)) | BDBM50446980 (CHEMBL3116048) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins University Curated by ChEMBL | Assay Description Inhibition of human recombinant GCP2 using N-acetyl-L-aspartyl[3H]-L-glutamate as substrate | J Med Chem 57: 243-7 (2014) Article DOI: 10.1021/jm401703a BindingDB Entry DOI: 10.7270/Q2HH6MJB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate carboxypeptidase 2 (Homo sapiens (Human)) | BDBM50446979 (CHEMBL3116049) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins University Curated by ChEMBL | Assay Description Inhibition of human recombinant GCP2 using N-acetyl-L-aspartyl[3H]-L-glutamate as substrate | J Med Chem 57: 243-7 (2014) Article DOI: 10.1021/jm401703a BindingDB Entry DOI: 10.7270/Q2HH6MJB | |||||||||||
More data for this Ligand-Target Pair |