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PubMed code 24389511

Compile data set for download or QSAR
Found 25 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Inhibitor of NF-kappa-B kinase (IKK)


(Homo sapiens (Human))
BDBM2579
PNG
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r|
Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1
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n/an/a 1n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of IKKbeta (unknown origin)


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
Tyrosine-protein kinase JAK2


(Homo sapiens (Human))
BDBM2579
PNG
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r|
Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1
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n/an/a 2n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of JAK2 (unknown origin)


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
Aurora kinase A


(Homo sapiens (Human))
BDBM2579
PNG
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r|
Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1
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n/an/a 15n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Aurora A (unknown origin)


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447157
PNG
(CHEMBL3112595)
Show SMILES CC(C)(C)NC(c1ccc(Cl)cc1)c1ccc(cc1)-c1cn[nH]c1
Show InChI InChI=1S/C20H22ClN3/c1-20(2,3)24-19(16-8-10-18(21)11-9-16)15-6-4-14(5-7-15)17-12-22-23-13-17/h4-13,19,24H,1-3H3,(H,22,23)
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n/an/a 38n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM2579
PNG
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r|
Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1
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n/an/a 40n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
Tyrosine-protein kinase SYK


(Homo sapiens (Human))
BDBM2579
PNG
((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Show SMILES CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r|
Show InChI InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1
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n/an/a 60n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of SYK (unknown origin)


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447174
PNG
(CHEMBL3113129)
Show SMILES CC(C)NC(c1ccc(Cl)cc1)c1ccc(cc1)-c1ncnc2nc[nH]c12
Show InChI InChI=1S/C21H20ClN5/c1-13(2)27-18(15-7-9-17(22)10-8-15)14-3-5-16(6-4-14)19-20-21(25-11-23-19)26-12-24-20/h3-13,18,27H,1-2H3,(H,23,24,25,26)
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n/an/a 160n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447170
PNG
(CHEMBL3113136)
Show SMILES CC(C)(C)NC(c1ccc(Cl)cc1)c1ccc(cc1)-c1ccncc1
Show InChI InChI=1S/C22H23ClN2/c1-22(2,3)25-21(19-8-10-20(23)11-9-19)18-6-4-16(5-7-18)17-12-14-24-15-13-17/h4-15,21,25H,1-3H3
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n/an/a 170n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447172
PNG
(CHEMBL3113134)
Show SMILES CC(C)NC(c1ccc(Cl)cc1)c1ccc(cc1)-c1ccncc1
Show InChI InChI=1S/C21H21ClN2/c1-15(2)24-21(19-7-9-20(22)10-8-19)18-5-3-16(4-6-18)17-11-13-23-14-12-17/h3-15,21,24H,1-2H3
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n/an/a 220n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447164
PNG
(CHEMBL3113143)
Show SMILES CC(C)NC(c1ccc(Cl)cc1)c1ccc(cc1)-c1cn[nH]c1
Show InChI InChI=1S/C19H20ClN3/c1-13(2)23-19(16-7-9-18(20)10-8-16)15-5-3-14(4-6-15)17-11-21-22-12-17/h3-13,19,23H,1-2H3,(H,21,22)
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n/an/a 370n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447173
PNG
(CHEMBL3113130)
Show SMILES Clc1ccc(cc1)C(NC1CC1)c1ccc(cc1)-c1ncnc2nc[nH]c12
Show InChI InChI=1S/C21H18ClN5/c22-16-7-5-14(6-8-16)18(27-17-9-10-17)13-1-3-15(4-2-13)19-20-21(25-11-23-19)26-12-24-20/h1-8,11-12,17-18,27H,9-10H2,(H,23,24,25,26)
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n/an/a 470n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447162
PNG
(CHEMBL3113145)
Show SMILES Clc1ccc(cc1)C(NC1CC1)c1ccc(cc1)-c1cn[nH]c1
Show InChI InChI=1S/C19H18ClN3/c20-17-7-5-15(6-8-17)19(23-18-9-10-18)14-3-1-13(2-4-14)16-11-21-22-12-16/h1-8,11-12,18-19,23H,9-10H2,(H,21,22)
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n/an/a 480n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447166
PNG
(CHEMBL3113141)
Show SMILES Clc1ccc(cc1)C(NC1CCCCC1)c1ccc(cc1)-c1ncnc2nc[nH]c12
Show InChI InChI=1S/C24H24ClN5/c25-19-12-10-17(11-13-19)21(30-20-4-2-1-3-5-20)16-6-8-18(9-7-16)22-23-24(28-14-26-22)29-15-27-23/h6-15,20-21,30H,1-5H2,(H,26,27,28,29)
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n/an/a 640n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447159
PNG
(CHEMBL3113149)
Show SMILES OCCNC(c1ccc(Cl)cc1)c1ccc(cc1)-c1cn[nH]c1
Show InChI InChI=1S/C18H18ClN3O/c19-17-7-5-15(6-8-17)18(20-9-10-23)14-3-1-13(2-4-14)16-11-21-22-12-16/h1-8,11-12,18,20,23H,9-10H2,(H,21,22)
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n/an/a 650n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447165
PNG
(CHEMBL3113142)
Show SMILES Clc1ccc(cc1)C(NCc1ccccc1)c1ccc(cc1)-c1ncnc2nc[nH]c12
Show InChI InChI=1S/C25H20ClN5/c26-21-12-10-19(11-13-21)22(27-14-17-4-2-1-3-5-17)18-6-8-20(9-7-18)23-24-25(30-15-28-23)31-16-29-24/h1-13,15-16,22,27H,14H2,(H,28,29,30,31)
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n/an/a 740n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447167
PNG
(CHEMBL3113140)
Show SMILES CC(C)CNC(c1ccc(Cl)cc1)c1ccc(cc1)-c1ncnc2nc[nH]c12
Show InChI InChI=1S/C22H22ClN5/c1-14(2)11-24-19(16-7-9-18(23)10-8-16)15-3-5-17(6-4-15)20-21-22(27-12-25-20)28-13-26-21/h3-10,12-14,19,24H,11H2,1-2H3,(H,25,26,27,28)
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n/an/a 740n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447158
PNG
(CHEMBL3113150)
Show SMILES NCCNC(c1ccc(Cl)cc1)c1ccc(cc1)-c1cn[nH]c1
Show InChI InChI=1S/C18H19ClN4/c19-17-7-5-15(6-8-17)18(21-10-9-20)14-3-1-13(2-4-14)16-11-22-23-12-16/h1-8,11-12,18,21H,9-10,20H2,(H,22,23)
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n/an/a 820n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAF serine/threonine protein kinase


(Homo sapiens (Human))
BDBM50447157
PNG
(CHEMBL3112595)
Show SMILES CC(C)(C)NC(c1ccc(Cl)cc1)c1ccc(cc1)-c1cn[nH]c1
Show InChI InChI=1S/C20H22ClN3/c1-20(2,3)24-19(16-8-10-18(21)11-9-16)15-6-4-14(5-7-15)17-12-22-23-13-17/h4-13,19,24H,1-3H3,(H,22,23)
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n/an/a 880n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of BRAF1 (unknown origin)


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447163
PNG
(CHEMBL3113144)
Show SMILES CC(C)CNC(c1ccc(Cl)cc1)c1ccc(cc1)-c1cn[nH]c1
Show InChI InChI=1S/C20H22ClN3/c1-14(2)11-22-20(17-7-9-19(21)10-8-17)16-5-3-15(4-6-16)18-12-23-24-13-18/h3-10,12-14,20,22H,11H2,1-2H3,(H,23,24)
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n/an/a 900n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447161
PNG
(CHEMBL3113146)
Show SMILES Clc1ccc(cc1)C(NC1CCCCC1)c1ccc(cc1)-c1cn[nH]c1
Show InChI InChI=1S/C22H24ClN3/c23-20-12-10-18(11-13-20)22(26-21-4-2-1-3-5-21)17-8-6-16(7-9-17)19-14-24-25-15-19/h6-15,21-22,26H,1-5H2,(H,24,25)
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n/an/a 1.10E+3n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447168
PNG
(CHEMBL3113139)
Show SMILES Clc1ccc(cc1)C(NCc1ccccc1)c1ccc(cc1)-c1ccncc1
Show InChI InChI=1S/C25H21ClN2/c26-24-12-10-23(11-13-24)25(28-18-19-4-2-1-3-5-19)22-8-6-20(7-9-22)21-14-16-27-17-15-21/h1-17,25,28H,18H2
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n/an/a 1.25E+3n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447169
PNG
(CHEMBL3113137)
Show SMILES Clc1ccc(cc1)C(NC1CCCCC1)c1ccc(cc1)-c1ccncc1
Show InChI InChI=1S/C24H25ClN2/c25-22-12-10-21(11-13-22)24(27-23-4-2-1-3-5-23)20-8-6-18(7-9-20)19-14-16-26-17-15-19/h6-17,23-24,27H,1-5H2
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n/an/a 1.26E+3n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447160
PNG
(CHEMBL3113148)
Show SMILES Clc1ccc(cc1)C(NCc1ccccc1)c1ccc(cc1)-c1cn[nH]c1
Show InChI InChI=1S/C23H20ClN3/c24-22-12-10-20(11-13-22)23(25-14-17-4-2-1-3-5-17)19-8-6-18(7-9-19)21-15-26-27-16-21/h1-13,15-16,23,25H,14H2,(H,26,27)
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n/an/a 1.32E+3n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM50447171
PNG
(CHEMBL3113135)
Show SMILES CC(C)CNC(c1ccc(Cl)cc1)c1ccc(cc1)-c1ccncc1
Show InChI InChI=1S/C22H23ClN2/c1-16(2)15-25-22(20-7-9-21(23)10-8-20)19-5-3-17(4-6-19)18-11-13-24-14-12-18/h3-14,16,22,25H,15H2,1-2H3
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n/an/a 1.43E+3n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase AKT1


(Homo sapiens (Human))
BDBM15211
PNG
(CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...)
Show SMILES Brc1ccc(\C=C\CNCCNS(=O)(=O)c2cccc3cnccc23)cc1
Show InChI InChI=1S/C20H20BrN3O2S/c21-18-8-6-16(7-9-18)3-2-11-22-13-14-24-27(25,26)20-5-1-4-17-15-23-12-10-19(17)20/h1-10,12,15,22,24H,11,13-14H2/b3-2+
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n/an/a 1.72E+3n/an/an/an/an/an/a



Zhejiang University

Curated by ChEMBL


Assay Description
Inhibition of Akt1 (unknown origin) using ATP/eNOS as substrate preincubated for 5 mins followed by substrate addition measured after 30 mins by fluo...


Eur J Med Chem 73: 167-76 (2014)


Article DOI: 10.1016/j.ejmech.2013.11.036
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%