Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50009298 (CHEMBL3233521) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Norwegian Medical Cyclotron Centre, PO Box 4950, Nydalen, N-0424 Oslo, Norway. Curated by ChEMBL | Assay Description Displacement of [125I]Triptorelin from rat full-length gonadotropin-releasing hormone receptor expressed in HEK293 cells | Bioorg Med Chem Lett 24: 1846-50 (2014) Article DOI: 10.1016/j.bmcl.2014.02.002 BindingDB Entry DOI: 10.7270/Q2XS5WXP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Mus musculus) | BDBM50261184 (5-((3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents | Article PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Norwegian Medical Cyclotron Centre, PO Box 4950, Nydalen, N-0424 Oslo, Norway. Curated by ChEMBL | Assay Description Binding affinity to mouse gonadotropin-releasing hormone receptor by radioligand displacement assay | Bioorg Med Chem Lett 24: 1846-50 (2014) Article DOI: 10.1016/j.bmcl.2014.02.002 BindingDB Entry DOI: 10.7270/Q2XS5WXP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50261184 (5-((3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents | Article PubMed | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Norwegian Medical Cyclotron Centre, PO Box 4950, Nydalen, N-0424 Oslo, Norway. Curated by ChEMBL | Assay Description Binding affinity to rat gonadotropin-releasing hormone receptor by radioligand displacement assay | Bioorg Med Chem Lett 24: 1846-50 (2014) Article DOI: 10.1016/j.bmcl.2014.02.002 BindingDB Entry DOI: 10.7270/Q2XS5WXP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50261184 (5-((3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphth...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Norwegian Medical Cyclotron Centre, PO Box 4950, Nydalen, N-0424 Oslo, Norway. Curated by ChEMBL | Assay Description Binding affinity to human gonadotropin-releasing hormone receptor by radioligand displacement assay | Bioorg Med Chem Lett 24: 1846-50 (2014) Article DOI: 10.1016/j.bmcl.2014.02.002 BindingDB Entry DOI: 10.7270/Q2XS5WXP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50224310 (5-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydro-naphth...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Norwegian Medical Cyclotron Centre, PO Box 4950, Nydalen, N-0424 Oslo, Norway. Curated by ChEMBL | Assay Description Binding affinity to human gonadotropin-releasing hormone receptor by radioligand displacement assay | Bioorg Med Chem Lett 24: 1846-50 (2014) Article DOI: 10.1016/j.bmcl.2014.02.002 BindingDB Entry DOI: 10.7270/Q2XS5WXP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50009297 (CHEMBL3233520) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 42 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Norwegian Medical Cyclotron Centre, PO Box 4950, Nydalen, N-0424 Oslo, Norway. Curated by ChEMBL | Assay Description Displacement of [125I]Triptorelin from rat full-length gonadotropin-releasing hormone receptor expressed in HEK293 cells | Bioorg Med Chem Lett 24: 1846-50 (2014) Article DOI: 10.1016/j.bmcl.2014.02.002 BindingDB Entry DOI: 10.7270/Q2XS5WXP | |||||||||||
More data for this Ligand-Target Pair |