Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
DNA helicase [35-727] (Plasmodium falciparum) | BDBM32017 ((7S,9S)-7-[(2R,4S,5S,6S)-4-azanyl-6-methyl-5-oxida...) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
International Centre for Genetic Engineering and Biotechnology | Assay Description Helicase assay was demonstrated using the purified fraction of PfUDN. The specially designed partial duplex substrate consisted of a 32P-labelled 47-... | BMC Biochem 15: 9 (2014) Article DOI: 10.1186/1471-2091-15-9 BindingDB Entry DOI: 10.7270/Q25H7F45 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA helicase [35-727] (Plasmodium falciparum) | BDBM200295 (AB00053825_07 | Ethidium bromide | cid_3624) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
International Centre for Genetic Engineering and Biotechnology | Assay Description The hydrolysis of ATP catalyzed by PfUDN was assayed by measuring the formation of Pi from [γ-32P] ATP. The reaction mixture of 10 μl conta... | BMC Biochem 15: 9 (2014) Article DOI: 10.1186/1471-2091-15-9 BindingDB Entry DOI: 10.7270/Q25H7F45 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA helicase [35-727] (Plasmodium falciparum) | BDBM50055660 (1-amino-3-(4-(4-(2-(amino(iminio)methylamino)aceta...) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL MMDB PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
International Centre for Genetic Engineering and Biotechnology | Assay Description The hydrolysis of ATP catalyzed by PfUDN was assayed by measuring the formation of Pi from [γ-32P] ATP. The reaction mixture of 10 μl conta... | BMC Biochem 15: 9 (2014) Article DOI: 10.1186/1471-2091-15-9 BindingDB Entry DOI: 10.7270/Q25H7F45 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA helicase [35-727] (Plasmodium falciparum) | BDBM50370548 (NOGALAMYCIN) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase MCE KEGG MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
International Centre for Genetic Engineering and Biotechnology | Assay Description The hydrolysis of ATP catalyzed by PfUDN was assayed by measuring the formation of Pi from [γ-32P] ATP. The reaction mixture of 10 μl conta... | BMC Biochem 15: 9 (2014) Article DOI: 10.1186/1471-2091-15-9 BindingDB Entry DOI: 10.7270/Q25H7F45 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA helicase [35-727] (Plasmodium falciparum) | BDBM50370548 (NOGALAMYCIN) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase MCE KEGG MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
International Centre for Genetic Engineering and Biotechnology | Assay Description Helicase assay was demonstrated using the purified fraction of PfUDN. The specially designed partial duplex substrate consisted of a 32P-labelled 47-... | BMC Biochem 15: 9 (2014) Article DOI: 10.1186/1471-2091-15-9 BindingDB Entry DOI: 10.7270/Q25H7F45 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA helicase [35-727] (Plasmodium falciparum) | BDBM32017 ((7S,9S)-7-[(2R,4S,5S,6S)-4-azanyl-6-methyl-5-oxida...) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 4.40E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
International Centre for Genetic Engineering and Biotechnology | Assay Description The hydrolysis of ATP catalyzed by PfUDN was assayed by measuring the formation of Pi from [γ-32P] ATP. The reaction mixture of 10 μl conta... | BMC Biochem 15: 9 (2014) Article DOI: 10.1186/1471-2091-15-9 BindingDB Entry DOI: 10.7270/Q25H7F45 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA helicase [35-727] (Plasmodium falciparum) | BDBM50055660 (1-amino-3-(4-(4-(2-(amino(iminio)methylamino)aceta...) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL MMDB PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
International Centre for Genetic Engineering and Biotechnology | Assay Description Helicase assay was demonstrated using the purified fraction of PfUDN. The specially designed partial duplex substrate consisted of a 32P-labelled 47-... | BMC Biochem 15: 9 (2014) Article DOI: 10.1186/1471-2091-15-9 BindingDB Entry DOI: 10.7270/Q25H7F45 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA helicase [35-727] (Plasmodium falciparum) | BDBM200295 (AB00053825_07 | Ethidium bromide | cid_3624) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
International Centre for Genetic Engineering and Biotechnology | Assay Description Helicase assay was demonstrated using the purified fraction of PfUDN. The specially designed partial duplex substrate consisted of a 32P-labelled 47-... | BMC Biochem 15: 9 (2014) Article DOI: 10.1186/1471-2091-15-9 BindingDB Entry DOI: 10.7270/Q25H7F45 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA helicase [35-727] (Plasmodium falciparum) | BDBM21690 (1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 9.90E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
International Centre for Genetic Engineering and Biotechnology | Assay Description The hydrolysis of ATP catalyzed by PfUDN was assayed by measuring the formation of Pi from [γ-32P] ATP. The reaction mixture of 10 μl conta... | BMC Biochem 15: 9 (2014) Article DOI: 10.1186/1471-2091-15-9 BindingDB Entry DOI: 10.7270/Q25H7F45 | |||||||||||
More data for this Ligand-Target Pair |