Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50442403 (CHEMBL494252) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Chungbuk National University Curated by ChEMBL | Assay Description Inhibition of porcine pancreatic lipase assessed as hydrolysis of p-NPB to p-nitrophenol by microplate reader | Bioorg Med Chem Lett 24: 2329-33 (2014) Article DOI: 10.1016/j.bmcl.2014.03.067 BindingDB Entry DOI: 10.7270/Q2V69M43 | |||||||||||
More data for this Ligand-Target Pair |