Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Deoxyribonuclease-1 (Homo sapiens (Human)) | BDBM50052802 (CHEBI:77181 | CRYSTAL VIOLET | Crystal violet (15)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nis Curated by ChEMBL | Assay Description Inhibition of DNase 1 (unknown origin) using (FAM)-labeled dsDNA as substrate | Eur J Med Chem 88: 101-11 (2014) Article DOI: 10.1016/j.ejmech.2014.07.040 BindingDB Entry DOI: 10.7270/Q2M32XC3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Deoxyribonuclease gamma (Homo sapiens (Human)) | BDBM50206432 (4-(4,6-dichloro-1,3,5-triazin-2-ylamino)-2-(6-hydr...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nis Curated by ChEMBL | Assay Description Inhibition of DNase gamma (unknown origin) transfected in HeLa S3 cells | Eur J Med Chem 88: 101-11 (2014) Article DOI: 10.1016/j.ejmech.2014.07.040 BindingDB Entry DOI: 10.7270/Q2M32XC3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Deoxyribonuclease-1 (Homo sapiens (Human)) | BDBM50206432 (4-(4,6-dichloro-1,3,5-triazin-2-ylamino)-2-(6-hydr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nis Curated by ChEMBL | Assay Description Inhibition of DNase 1 (unknown origin) | Eur J Med Chem 88: 101-11 (2014) Article DOI: 10.1016/j.ejmech.2014.07.040 BindingDB Entry DOI: 10.7270/Q2M32XC3 | |||||||||||
More data for this Ligand-Target Pair |