Found 22 hits of Enzyme Inhibition Constant Data Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055195
(CHEMBL3323612)Show SMILES Clc1ccc(cc1Cl)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H14Cl2N4/c23-16-7-5-13(11-17(16)24)22-27-20-8-6-14(12-21(20)28-22)26-19-9-10-25-18-4-2-1-3-15(18)19/h1-12H,(H,25,26)(H,27,28) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM4814
(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)Show SMILES CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C Show InChI InChI=1S/C22H27FN4O2/c1-5-27(6-2)10-9-24-22(29)20-13(3)19(25-14(20)4)12-17-16-11-15(23)7-8-18(16)26-21(17)28/h7-8,11-12,25H,5-6,9-10H2,1-4H3,(H,24,29)(H,26,28)/b17-12- | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
DrugBank
MCE
MMDB
PC cid
PC sid
PDB
UniChem
Patents
Similars
| DrugBank
PDB
Article
PubMed
| n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | 
3D Structure (crystal) |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055215
(CHEMBL3323613)Show SMILES Clc1cc(Cl)cc(c1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H14Cl2N4/c23-14-9-13(10-15(24)11-14)22-27-20-6-5-16(12-21(20)28-22)26-19-7-8-25-18-4-2-1-3-17(18)19/h1-12H,(H,25,26)(H,27,28) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055158
(CHEMBL3323605)Show SMILES Brc1ccc(cc1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H15BrN4/c23-15-7-5-14(6-8-15)22-26-20-10-9-16(13-21(20)27-22)25-19-11-12-24-18-4-2-1-3-17(18)19/h1-13H,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055155
(CHEMBL3323604)Show SMILES Clc1ccc(cc1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H15ClN4/c23-15-7-5-14(6-8-15)22-26-20-10-9-16(13-21(20)27-22)25-19-11-12-24-18-4-2-1-3-17(18)19/h1-13H,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055110
(CHEMBL3323601)Show SMILES Fc1ccc(cc1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H15FN4/c23-15-7-5-14(6-8-15)22-26-20-10-9-16(13-21(20)27-22)25-19-11-12-24-18-4-2-1-3-17(18)19/h1-13H,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.36E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055144
(CHEMBL3323603)Show SMILES Clc1cccc(c1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H15ClN4/c23-15-5-3-4-14(12-15)22-26-20-9-8-16(13-21(20)27-22)25-19-10-11-24-18-7-2-1-6-17(18)19/h1-13H,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055101
(CHEMBL3323592)Show SMILES N(c1ccc2nc([nH]c2c1)-c1ccccc1)c1ccnc2ccccc12 Show InChI InChI=1S/C22H16N4/c1-2-6-15(7-3-1)22-25-20-11-10-16(14-21(20)26-22)24-19-12-13-23-18-9-5-4-8-17(18)19/h1-14H,(H,23,24)(H,25,26) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 2.48E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055109
(CHEMBL3323600)Show SMILES Fc1cccc(c1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H15FN4/c23-15-5-3-4-14(12-15)22-26-20-9-8-16(13-21(20)27-22)25-19-10-11-24-18-7-2-1-6-17(18)19/h1-13H,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 3.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055104
(CHEMBL3323595)Show SMILES Cc1ccc(cc1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C23H18N4/c1-15-6-8-16(9-7-15)23-26-21-11-10-17(14-22(21)27-23)25-20-12-13-24-19-5-3-2-4-18(19)20/h2-14H,1H3,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 4.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055107
(CHEMBL3323598)Show SMILES CCc1ccc(cc1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C24H20N4/c1-2-16-7-9-17(10-8-16)24-27-22-12-11-18(15-23(22)28-24)26-21-13-14-25-20-6-4-3-5-19(20)21/h3-15H,2H2,1H3,(H,25,26)(H,27,28) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 5.49E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055103
(CHEMBL3323594)Show SMILES Cc1cccc(c1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C23H18N4/c1-15-5-4-6-16(13-15)23-26-21-10-9-17(14-22(21)27-23)25-20-11-12-24-19-8-3-2-7-18(19)20/h2-14H,1H3,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055221
(CHEMBL3323614)Show SMILES Fc1ccc(Br)c(c1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H14BrFN4/c23-17-7-5-13(24)11-16(17)22-27-20-8-6-14(12-21(20)28-22)26-19-9-10-25-18-4-2-1-3-15(18)19/h1-12H,(H,25,26)(H,27,28) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 7.82E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055191
(CHEMBL3323611)Show SMILES Clc1cccc(Cl)c1-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H14Cl2N4/c23-15-5-3-6-16(24)21(15)22-27-19-9-8-13(12-20(19)28-22)26-18-10-11-25-17-7-2-1-4-14(17)18/h1-12H,(H,25,26)(H,27,28) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
MMDB
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| n/a | n/a | 8.35E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055106
(CHEMBL3323597)Show SMILES Oc1ccccc1-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H16N4O/c27-21-8-4-2-6-16(21)22-25-19-10-9-14(13-20(19)26-22)24-18-11-12-23-17-7-3-1-5-15(17)18/h1-13,27H,(H,23,24)(H,25,26) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 9.53E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055177
(CHEMBL3323609)Show SMILES FC(F)(F)c1cccc(c1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C23H15F3N4/c24-23(25,26)15-5-3-4-14(12-15)22-29-20-9-8-16(13-21(20)30-22)28-19-10-11-27-18-7-2-1-6-17(18)19/h1-13H,(H,27,28)(H,29,30) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055108
(CHEMBL3323599)Show SMILES Fc1ccccc1-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H15FN4/c23-17-7-3-1-5-15(17)22-26-20-10-9-14(13-21(20)27-22)25-19-11-12-24-18-8-4-2-6-16(18)19/h1-13H,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055105
(CHEMBL3323596)Show SMILES COc1ccccc1-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C23H18N4O/c1-28-22-9-5-3-7-17(22)23-26-20-11-10-15(14-21(20)27-23)25-19-12-13-24-18-8-4-2-6-16(18)19/h2-14H,1H3,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055174
(CHEMBL3323606)Show SMILES FC(F)(F)c1ccccc1-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C23H15F3N4/c24-23(25,26)17-7-3-1-5-15(17)22-29-20-10-9-14(13-21(20)30-22)28-19-11-12-27-18-8-4-2-6-16(18)19/h1-13H,(H,27,28)(H,29,30) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055102
(CHEMBL3323593)Show SMILES Cc1ccccc1-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C23H18N4/c1-15-6-2-3-7-17(15)23-26-21-11-10-16(14-22(21)27-23)25-20-12-13-24-19-9-5-4-8-18(19)20/h2-14H,1H3,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055111
(CHEMBL3323602)Show SMILES Clc1ccccc1-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C22H15ClN4/c23-17-7-3-1-5-15(17)22-26-20-10-9-14(13-21(20)27-22)25-19-11-12-24-18-8-4-2-6-16(18)19/h1-13H,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50055182
(CHEMBL3323610)Show SMILES FC(F)(F)c1ccc(cc1)-c1nc2ccc(Nc3ccnc4ccccc34)cc2[nH]1 Show InChI InChI=1S/C23H15F3N4/c24-23(25,26)15-7-5-14(6-8-15)22-29-20-10-9-16(13-21(20)30-22)28-19-11-12-27-18-4-2-1-3-17(18)19/h1-13H,(H,27,28)(H,29,30) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University
Curated by ChEMBL
| Assay Description
Inhibition of VEGFR2 (unknown origin) using ATP/substrate peptide after 1 hr by colorimetric ELISA |
Eur J Med Chem 84: 698-707 (2014)
Article DOI: 10.1016/j.ejmech.2014.07.071
BindingDB Entry DOI: 10.7270/Q26Q1ZWB |
More data for this
Ligand-Target Pair | |
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