Affinity Data by PubMed id=25082125

PubMed code 25082125

Found 12 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cytochrome P450 2C9 (Homo sapiens (Human))	BDBM50100544 (CHEMBL3321835) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.69E+4	n/a	n/a	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Inhibition of CYP2C9 (unknown origin)				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100549 (CHEMBL3321831) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	173	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100551 (CHEMBL3321829) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	240	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100552 (CHEMBL3321828) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	100	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100554 (CHEMBL3321827) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100555 (CHEMBL3321826) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	39	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100545 (CHEMBL3321838) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	140	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100548 (CHEMBL3321832) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	781	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100550 (CHEMBL3321830) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	82	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100544 (CHEMBL3321835) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	3	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100547 (CHEMBL3321834) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50100546 (CHEMBL3321837) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	26	n/a	n/a	n/a	n/a
Korea Research Institute of Chemical Technology Curated by ChEMBL					Assay Description Agonist activity at human GPR119 expressed in CHO-K1 cells after 24 hrs by CRE-luciferase assay				Bioorg Med Chem Lett 24: 4281-5 (2014) Article DOI: 10.1016/j.bmcl.2014.07.020 BindingDB Entry DOI: 10.7270/Q29S1SSJ
					More data for this Ligand-Target Pair

* indicates data uncertainty>20%