Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proto-oncogene tyrosine-protein kinase Src (Homo sapiens (Human)) | BDBM150751 (CPR005231 (6)) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | 7.5 | 25 |
University of Copenhagen | Assay Description The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b... | Chembiochem 16: 59-63 (2015) Article DOI: 10.1002/cbic.201402512 BindingDB Entry DOI: 10.7270/Q2XW4HHD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Death-associated protein kinase 1 (Homo sapiens (Human)) | BDBM150751 (CPR005231 (6)) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 247 | n/a | n/a | n/a | n/a | 7.5 | 25 |
University of Copenhagen | Assay Description The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b... | Chembiochem 16: 59-63 (2015) Article DOI: 10.1002/cbic.201402512 BindingDB Entry DOI: 10.7270/Q2XW4HHD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human)) | BDBM150751 (CPR005231 (6)) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | 7.5 | 25 |
University of Copenhagen | Assay Description The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b... | Chembiochem 16: 59-63 (2015) Article DOI: 10.1002/cbic.201402512 BindingDB Entry DOI: 10.7270/Q2XW4HHD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK2 (Homo sapiens (Human)) | BDBM150751 (CPR005231 (6)) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | 7.5 | 25 |
University of Copenhagen | Assay Description The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b... | Chembiochem 16: 59-63 (2015) Article DOI: 10.1002/cbic.201402512 BindingDB Entry DOI: 10.7270/Q2XW4HHD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase PAK 5 (Homo sapiens (Human)) | BDBM150751 (CPR005231 (6)) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.60E+3 | n/a | n/a | n/a | n/a | 7.5 | 25 |
University of Copenhagen | Assay Description The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b... | Chembiochem 16: 59-63 (2015) Article DOI: 10.1002/cbic.201402512 BindingDB Entry DOI: 10.7270/Q2XW4HHD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Death-associated protein kinase 1 (Homo sapiens (Human)) | BDBM150751 (CPR005231 (6)) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 240 | n/a | n/a | n/a | 7.5 | n/a |
University of Copenhagen | Assay Description 40 µL of a solution containing 350-500 µM of CPR005231 (compound 6) were titrated into the 200 µL sample cell containing 25-55 µM DAPK1 (AA 1-285) or... | Chembiochem 16: 59-63 (2015) Article DOI: 10.1002/cbic.201402512 BindingDB Entry DOI: 10.7270/Q2XW4HHD | |||||||||||
More data for this Ligand-Target Pair |