Found 45 hits of Enzyme Inhibition Constant Data Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095454
(CHEMBL3590422)Show InChI InChI=1S/C15H30N2O4/c1-3-4-11-16(2)12-8-6-5-7-9-14(18)17(21)13-10-15(19)20/h21H,3-13H2,1-2H3,(H,19,20) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095446
(CHEMBL3590426)Show InChI InChI=1S/C14H28N2O4/c1-3-4-6-10-15(2)11-7-5-8-13(17)16(20)12-9-14(18)19/h20H,3-12H2,1-2H3,(H,18,19) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095451
(CHEMBL3590431)Show InChI InChI=1S/C20H40N2O4/c1-3-5-7-8-9-11-16-21(15-6-4-2)17-12-10-13-19(23)22(26)18-14-20(24)25/h26H,3-18H2,1-2H3,(H,24,25) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095447
(CHEMBL3590427)Show InChI InChI=1S/C15H30N2O4/c1-3-4-5-7-11-16(2)12-8-6-9-14(18)17(21)13-10-15(19)20/h21H,3-13H2,1-2H3,(H,19,20) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095445
(CHEMBL3590421)Show InChI InChI=1S/C14H28N2O4/c1-3-4-10-15(2)11-7-5-6-8-13(17)16(20)12-9-14(18)19/h20H,3-12H2,1-2H3,(H,18,19) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095443
(CHEMBL3590418)Show InChI InChI=1S/C13H26N2O4/c1-3-4-9-14(2)10-6-5-7-12(16)15(19)11-8-13(17)18/h19H,3-11H2,1-2H3,(H,17,18) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 4.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095448
(CHEMBL3590430)Show InChI InChI=1S/C18H36N2O4/c1-3-5-7-9-14-19(13-6-4-2)15-10-8-11-17(21)20(24)16-12-18(22)23/h24H,3-16H2,1-2H3,(H,22,23) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 4.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095453
(CHEMBL3590420)Show InChI InChI=1S/C12H24N2O4/c1-3-4-8-13(2)9-5-6-11(15)14(18)10-7-12(16)17/h18H,3-10H2,1-2H3,(H,16,17) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 6.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095454
(CHEMBL3590422)Show InChI InChI=1S/C15H30N2O4/c1-3-4-11-16(2)12-8-6-5-7-9-14(18)17(21)13-10-15(19)20/h21H,3-13H2,1-2H3,(H,19,20) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 6.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095456
(CHEMBL3590424)Show InChI InChI=1S/C11H22N2O4/c1-3-12(2)8-5-4-6-10(14)13(17)9-7-11(15)16/h17H,3-9H2,1-2H3,(H,15,16) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 7.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095457
(CHEMBL3590425)Show InChI InChI=1S/C12H24N2O4/c1-3-8-13(2)9-5-4-6-11(15)14(18)10-7-12(16)17/h18H,3-10H2,1-2H3,(H,16,17) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 8.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095458
(CHEMBL3590428)Show InChI InChI=1S/C14H28N2O4/c1-3-5-10-15(4-2)11-7-6-8-13(17)16(20)12-9-14(18)19/h20H,3-12H2,1-2H3,(H,18,19) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095455
(CHEMBL3590423)Show InChI InChI=1S/C10H20N2O4/c1-11(2)7-4-3-5-9(13)12(16)8-6-10(14)15/h16H,3-8H2,1-2H3,(H,14,15) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095459
(CHEMBL3590429)Show InChI InChI=1S/C16H32N2O4/c1-3-5-11-17(12-6-4-2)13-8-7-9-15(19)18(22)14-10-16(20)21/h22H,3-14H2,1-2H3,(H,20,21) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095461
(CHEMBL3590433)Show InChI InChI=1S/C16H32N2O4/c1-4-5-6-8-12-17(2)13-9-7-10-15(19)18(21)14-11-16(20)22-3/h21H,4-14H2,1-3H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Histone lysine demethylase PHF8
(Homo sapiens (Human)) | BDBM50095451
(CHEMBL3590431)Show InChI InChI=1S/C20H40N2O4/c1-3-5-7-8-9-11-16-21(15-6-4-2)17-12-10-13-19(23)22(26)18-14-20(24)25/h26H,3-18H2,1-2H3,(H,24,25) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JHDM1F (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Histone lysine demethylase PHF8
(Homo sapiens (Human)) | BDBM50095448
(CHEMBL3590430)Show InChI InChI=1S/C18H36N2O4/c1-3-5-7-9-14-19(13-6-4-2)15-10-8-11-17(21)20(24)16-12-18(22)23/h24H,3-16H2,1-2H3,(H,22,23) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 2.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JHDM1F (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095446
(CHEMBL3590426)Show InChI InChI=1S/C14H28N2O4/c1-3-4-6-10-15(2)11-7-5-8-13(17)16(20)12-9-14(18)19/h20H,3-12H2,1-2H3,(H,18,19) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 3.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095447
(CHEMBL3590427)Show InChI InChI=1S/C15H30N2O4/c1-3-4-5-7-11-16(2)12-8-6-9-14(18)17(21)13-10-15(19)20/h21H,3-13H2,1-2H3,(H,19,20) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 4.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095455
(CHEMBL3590423)Show InChI InChI=1S/C10H20N2O4/c1-11(2)7-4-3-5-9(13)12(16)8-6-10(14)15/h16H,3-8H2,1-2H3,(H,14,15) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 5.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095452
(CHEMBL3590419)Show InChI InChI=1S/C11H22N2O4/c1-3-4-7-12(2)8-5-10(14)13(17)9-6-11(15)16/h17H,3-9H2,1-2H3,(H,15,16) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 5.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095443
(CHEMBL3590418)Show InChI InChI=1S/C13H26N2O4/c1-3-4-9-14(2)10-6-5-7-12(16)15(19)11-8-13(17)18/h19H,3-11H2,1-2H3,(H,17,18) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 5.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Histone lysine demethylase PHF8
(Homo sapiens (Human)) | BDBM50095445
(CHEMBL3590421)Show InChI InChI=1S/C14H28N2O4/c1-3-4-10-15(2)11-7-5-6-8-13(17)16(20)12-9-14(18)19/h20H,3-12H2,1-2H3,(H,18,19) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 5.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JHDM1F (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095445
(CHEMBL3590421)Show InChI InChI=1S/C14H28N2O4/c1-3-4-10-15(2)11-7-5-6-8-13(17)16(20)12-9-14(18)19/h20H,3-12H2,1-2H3,(H,18,19) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 6.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095456
(CHEMBL3590424)Show InChI InChI=1S/C11H22N2O4/c1-3-12(2)8-5-4-6-10(14)13(17)9-7-11(15)16/h17H,3-9H2,1-2H3,(H,15,16) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 6.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM50095460
(CHEMBL3590432)Show InChI InChI=1S/C15H30N2O4/c1-4-5-7-11-16(2)12-8-6-9-14(18)17(20)13-10-15(19)21-3/h20H,4-13H2,1-3H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 6.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095453
(CHEMBL3590420)Show InChI InChI=1S/C12H24N2O4/c1-3-4-8-13(2)9-5-6-11(15)14(18)10-7-12(16)17/h18H,3-10H2,1-2H3,(H,16,17) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 6.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095458
(CHEMBL3590428)Show InChI InChI=1S/C14H28N2O4/c1-3-5-10-15(4-2)11-7-6-8-13(17)16(20)12-9-14(18)19/h20H,3-12H2,1-2H3,(H,18,19) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 6.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Histone lysine demethylase PHF8
(Homo sapiens (Human)) | BDBM50095447
(CHEMBL3590427)Show InChI InChI=1S/C15H30N2O4/c1-3-4-5-7-11-16(2)12-8-6-9-14(18)17(21)13-10-15(19)20/h21H,3-13H2,1-2H3,(H,19,20) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 7.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JHDM1F (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095457
(CHEMBL3590425)Show InChI InChI=1S/C12H24N2O4/c1-3-8-13(2)9-5-4-6-11(15)14(18)10-7-12(16)17/h18H,3-10H2,1-2H3,(H,16,17) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 7.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095451
(CHEMBL3590431)Show InChI InChI=1S/C20H40N2O4/c1-3-5-7-8-9-11-16-21(15-6-4-2)17-12-10-13-19(23)22(26)18-14-20(24)25/h26H,3-18H2,1-2H3,(H,24,25) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 8.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 3A
(Homo sapiens (Human)) | BDBM50095443
(CHEMBL3590418)Show InChI InChI=1S/C13H26N2O4/c1-3-4-9-14(2)10-6-5-7-12(16)15(19)11-8-13(17)18/h19H,3-11H2,1-2H3,(H,17,18) | Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD1A (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 3A
(Homo sapiens (Human)) | BDBM50095447
(CHEMBL3590427)Show InChI InChI=1S/C15H30N2O4/c1-3-4-5-7-11-16(2)12-8-6-9-14(18)17(21)13-10-15(19)20/h21H,3-13H2,1-2H3,(H,19,20) | Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD1A (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 3A
(Homo sapiens (Human)) | BDBM50095451
(CHEMBL3590431)Show InChI InChI=1S/C20H40N2O4/c1-3-5-7-8-9-11-16-21(15-6-4-2)17-12-10-13-19(23)22(26)18-14-20(24)25/h26H,3-18H2,1-2H3,(H,24,25) | Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD1A (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095452
(CHEMBL3590419)Show InChI InChI=1S/C11H22N2O4/c1-3-4-7-12(2)8-5-10(14)13(17)9-6-11(15)16/h17H,3-9H2,1-2H3,(H,15,16) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095459
(CHEMBL3590429)Show InChI InChI=1S/C16H32N2O4/c1-3-5-11-17(12-6-4-2)13-8-7-9-15(19)18(22)14-10-16(20)21/h22H,3-14H2,1-2H3,(H,20,21) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM50095448
(CHEMBL3590430)Show InChI InChI=1S/C18H36N2O4/c1-3-5-7-9-14-19(13-6-4-2)15-10-8-11-17(21)20(24)16-12-18(22)23/h24H,3-16H2,1-2H3,(H,22,23) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 3A
(Homo sapiens (Human)) | BDBM50095448
(CHEMBL3590430)Show InChI InChI=1S/C18H36N2O4/c1-3-5-7-9-14-19(13-6-4-2)15-10-8-11-17(21)20(24)16-12-18(22)23/h24H,3-16H2,1-2H3,(H,22,23) | Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD1A (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Histone lysine demethylase PHF8
(Homo sapiens (Human)) | BDBM50095446
(CHEMBL3590426)Show InChI InChI=1S/C14H28N2O4/c1-3-4-6-10-15(2)11-7-5-8-13(17)16(20)12-9-14(18)19/h20H,3-12H2,1-2H3,(H,18,19) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JHDM1F (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Histone lysine demethylase PHF8
(Homo sapiens (Human)) | BDBM50095443
(CHEMBL3590418)Show InChI InChI=1S/C13H26N2O4/c1-3-4-9-14(2)10-6-5-7-12(16)15(19)11-8-13(17)18/h19H,3-11H2,1-2H3,(H,17,18) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JHDM1F (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 3A
(Homo sapiens (Human)) | BDBM50095446
(CHEMBL3590426)Show InChI InChI=1S/C14H28N2O4/c1-3-4-6-10-15(2)11-7-5-8-13(17)16(20)12-9-14(18)19/h20H,3-12H2,1-2H3,(H,18,19) | Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD1A (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 5A
(Homo sapiens (Human)) | BDBM26106
(CHEMBL90852 | N-oxalyl glycine, 1a | NOG | Oxalylg...)Show InChI InChI=1S/C4H5NO5/c6-2(7)1-5-3(8)4(9)10/h1H2,(H,5,8)(H,6,7)(H,9,10) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE MMDB PC cid PC sid PDB UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Lysine-specific demethylase 4C
(Homo sapiens (Human)) | BDBM26106
(CHEMBL90852 | N-oxalyl glycine, 1a | NOG | Oxalylg...)Show InChI InChI=1S/C4H5NO5/c6-2(7)1-5-3(8)4(9)10/h1H2,(H,5,8)(H,6,7)(H,9,10) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PDB Article PubMed
| n/a | n/a | 4.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD2C (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | 3D Structure (crystal) |
Lysine-specific demethylase 3A
(Homo sapiens (Human)) | BDBM26106
(CHEMBL90852 | N-oxalyl glycine, 1a | NOG | Oxalylg...)Show InChI InChI=1S/C4H5NO5/c6-2(7)1-5-3(8)4(9)10/h1H2,(H,5,8)(H,6,7)(H,9,10) | Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE MMDB PC cid PC sid PDB UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 5.69E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JMJD1A (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | |
Histone lysine demethylase PHF8
(Homo sapiens (Human)) | BDBM26106
(CHEMBL90852 | N-oxalyl glycine, 1a | NOG | Oxalylg...)Show InChI InChI=1S/C4H5NO5/c6-2(7)1-5-3(8)4(9)10/h1H2,(H,5,8)(H,6,7)(H,9,10) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE MMDB PC cid PC sid PDB UniChem
Patents
Similars
| PDB Article PubMed
| n/a | n/a | 6.40E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University of Medicine
Curated by ChEMBL
| Assay Description Inhibition of JHDM1F (unknown origin) using H3K9mel peptide |
ACS Med Chem Lett 6: 665-70 (2015)
Article DOI: 10.1021/acsmedchemlett.5b00083 BindingDB Entry DOI: 10.7270/Q2V69MC7 |
More data for this Ligand-Target Pair | 3D Structure (crystal) |