Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50115191 (CHEMBL3609573) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 510 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRalpha expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubate... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50115191 (CHEMBL3609573) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 160 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRbeta expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubated... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50115193 (CHEMBL3609363) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 260 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRbeta expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubated... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50115195 (CHEMBL3609361) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRbeta expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubated... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50115195 (CHEMBL3609361) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 540 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRalpha expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubate... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50115194 (CHEMBL3609362) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 310 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRalpha expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubate... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM19993 (CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRalpha expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubate... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50115194 (CHEMBL3609362) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 210 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRbeta expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubated... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50115192 (CHEMBL3609572) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRalpha expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubate... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM19993 (CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 130 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRbeta expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubated... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50115192 (CHEMBL3609572) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 530 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRbeta expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubated... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50115193 (CHEMBL3609363) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 280 | n/a | n/a | n/a | n/a |
Daiichi Sankyo RD Novare Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human LXRalpha expressed in African green monkey kidney CV1 cells co-expressing pTAL-LXRE including LXR response element incubate... | Bioorg Med Chem Lett 25: 3914-20 (2015) Article DOI: 10.1016/j.bmcl.2015.07.047 BindingDB Entry DOI: 10.7270/Q23T9K08 | |||||||||||
More data for this Ligand-Target Pair |