Affinity Data by PubMed id=26928019

PubMed code 26928019

Found 39 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157567 (CHEMBL3785789) Show SMILES CCCCCCCC#Cc1ccc(CCC(O)=O)cc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	1.45E+3	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157619 (CHEMBL3787072) Show SMILES C\C=C/C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	48	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50275510 (3-(4-(Phenylethynyl)phenyl)propanoic acid \| CHEMBL...) Show SMILES OC(=O)CCc1ccc(cc1)C#Cc1ccccc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	8.51E+3	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157602 (CHEMBL3787165) Show SMILES OC(=O)CCc1ccc(cc1)C#CC1(O)CCCCC1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	<1.00E+5	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157614 (CHEMBL3786972) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	7.59E+3	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157617 (CHEMBL3785764) Show SMILES C\C=C(/C)C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.63E+4	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157619 (CHEMBL3787072) Show SMILES C\C=C/C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.78E+4	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157620 (CHEMBL3785413) Show SMILES C\C(=C\CO)C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	<1.00E+5	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157571 (CHEMBL3786964) Show SMILES OC(=O)CCc1ccc(cc1)C#CC1CC1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	5.01E+3	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157600 (CHEMBL3787110) Show SMILES OC(=O)CCc1ccc(cc1)C#CC1CCCC1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	490	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157613 (CHEMBL3785544) Show SMILES CC(=C)C#Cc1ccc(CCC(O)=O)cc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	417	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157617 (CHEMBL3785764) Show SMILES C\C=C(/C)C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	37	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157566 (CHEMBL3785667) Show SMILES OC(=O)CCc1ccc(cc1)C#C Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	<1.00E+5	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157568 (CHEMBL3787580) Show SMILES OC(=O)CCc1ccc(cc1)C#CCc1ccccc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	1.05E+4	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157613 (CHEMBL3785544) Show SMILES CC(=C)C#Cc1ccc(CCC(O)=O)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	<1.00E+5	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157566 (CHEMBL3785667) Show SMILES OC(=O)CCc1ccc(cc1)C#C Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	<1.00E+5	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157568 (CHEMBL3787580) Show SMILES OC(=O)CCc1ccc(cc1)C#CCc1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	389	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157618 (CHEMBL3785637) Show SMILES C\C=C(\C)C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	20	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157567 (CHEMBL3785789) Show SMILES CCCCCCCC#Cc1ccc(CCC(O)=O)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	4.07E+3	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157616 (CHEMBL3786526) Show SMILES C\C=C\C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	3.47E+4	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157603 (CHEMBL3786524) Show SMILES OC(=O)CCc1ccc(cc1)C#CC1=CCCCC1 \|t:14\| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	200	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157618 (CHEMBL3785637) Show SMILES C\C=C(\C)C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	20	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157620 (CHEMBL3785413) Show SMILES C\C(=C\CO)C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	427	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157615 (CHEMBL3787463) Show SMILES CC(=C)C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	n/a	n/a	<1.00E+5	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50240347 ((9,12,15)-linolenic acid \| (9Z,12Z,15Z)-octadeca-9...) Show SMILES CC\C=C/C\C=C/C\C=C/CCCCCCCC(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	3.16E+3	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157601 (CHEMBL3786418) Show SMILES OC(=O)CCc1ccc(cc1)C#CC1CCCCC1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	513	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157602 (CHEMBL3787165) Show SMILES OC(=O)CCc1ccc(cc1)C#CC1(O)CCCCC1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50240347 ((9,12,15)-linolenic acid \| (9Z,12Z,15Z)-octadeca-9...) Show SMILES CC\C=C/C\C=C/C\C=C/CCCCCCCC(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	3.00E+3	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157569 (CHEMBL3787151) Show SMILES OC(=O)CCc1ccc(cc1)C#CCCc1ccccc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	4.79E+3	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157600 (CHEMBL3787110) Show SMILES OC(=O)CCc1ccc(cc1)C#CC1CCCC1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	3.39E+4	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157615 (CHEMBL3787463) Show SMILES CC(=C)C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	n/a	n/a	81	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157601 (CHEMBL3786418) Show SMILES OC(=O)CCc1ccc(cc1)C#CC1CCCCC1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	9.55E+3	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157603 (CHEMBL3786524) Show SMILES OC(=O)CCc1ccc(cc1)C#CC1=CCCCC1 \|t:14\| Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<1.00E+5	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157614 (CHEMBL3786972) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	83	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157571 (CHEMBL3786964) Show SMILES OC(=O)CCc1ccc(cc1)C#CC1CC1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	<1.00E+5	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50157618 (CHEMBL3785637) Show SMILES C\C=C(\C)C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.00E+4	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50275510 (3-(4-(Phenylethynyl)phenyl)propanoic acid \| CHEMBL...) Show SMILES OC(=O)CCc1ccc(cc1)C#Cc1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	200	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157616 (CHEMBL3786526) Show SMILES C\C=C\C#Cc1ccc(CCC(O)=O)c(F)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	209	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 1 (Homo sapiens (Human))	BDBM50157569 (CHEMBL3787151) Show SMILES OC(=O)CCc1ccc(cc1)C#CCCc1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	1.82E+3	n/a	n/a	n/a	n/a
University of Southern Denmark Curated by ChEMBL					Assay Description Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay				J Med Chem 59: 2841-6 (2016) Article DOI: 10.1021/acs.jmedchem.5b01962 BindingDB Entry DOI: 10.7270/Q2PN97HD
University of Southern Denmark Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%