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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM181101 (N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet  | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM181097 (N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.72E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM181098 (N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Insulin receptor (Homo sapiens (Human)) | BDBM181101 (N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Vascular endothelial growth factor receptor 1 (Homo sapiens (Human)) | BDBM181101 (N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Fibroblast growth factor receptor 1 (Homo sapiens (Human)) | BDBM181098 (N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Vascular endothelial growth factor receptor 1 (Homo sapiens (Human)) | BDBM181097 (N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM181095 (N-(4-Hydroxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM181099 (N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.15E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Fibroblast growth factor receptor 1 (Homo sapiens (Human)) | BDBM181101 (N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Insulin receptor (Homo sapiens (Human)) | BDBM181097 (N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.26E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Fibroblast growth factor receptor 1 (Homo sapiens (Human)) | BDBM181097 (N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.29E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Vascular endothelial growth factor receptor 1 (Homo sapiens (Human)) | BDBM181098 (N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.29E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Insulin receptor (Homo sapiens (Human)) | BDBM181098 (N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.76E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM181096 (N-(4-fluorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM181100 (N-(4-Trifluoromethylbenzylidene)-2-(3,6-dimethyl-1...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.59E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Beni-Suef University | Assay Description Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t... | Bioorg Chem 66: 88-96 (2016) Article DOI: 10.1016/j.bioorg.2016.03.011 BindingDB Entry DOI: 10.7270/Q2VQ31GF | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
