Found 10 hits of Enzyme Inhibition Constant Data Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Serine/threonine-protein kinase 16
(Homo sapiens (Human)) | BDBM185152
(STK16-IN-1)Show InChI InChI=1S/C16H10FN3O2/c17-12-3-2-10(7-13(12)21)20-14(22)4-1-9-8-19-16-11(15(9)20)5-6-18-16/h1-8,21H,(H,18,19) | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 295 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences
| Assay Description
The enzymatic assay was performed using the LifeTechnology SelectScreen. |
ACS Chem Biol 11: 1537-43 (2016)
Article DOI: 10.1021/acschembio.6b00250
BindingDB Entry DOI: 10.7270/Q29K491Z |
More data for this
Ligand-Target Pair | |
Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform
(Homo sapiens (Human)) | BDBM185152
(STK16-IN-1)Show InChI InChI=1S/C16H10FN3O2/c17-12-3-2-10(7-13(12)21)20-14(22)4-1-9-8-19-16-11(15(9)20)5-6-18-16/h1-8,21H,(H,18,19) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 856 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences
| Assay Description
The enzymatic assay was performed using the LifeTechnology SelectScreen. |
ACS Chem Biol 11: 1537-43 (2016)
Article DOI: 10.1021/acschembio.6b00250
BindingDB Entry DOI: 10.7270/Q29K491Z |
More data for this
Ligand-Target Pair | |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
(Homo sapiens (Human)) | BDBM185152
(STK16-IN-1)Show InChI InChI=1S/C16H10FN3O2/c17-12-3-2-10(7-13(12)21)20-14(22)4-1-9-8-19-16-11(15(9)20)5-6-18-16/h1-8,21H,(H,18,19) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 867 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences
| Assay Description
The enzymatic assay was performed using the LifeTechnology SelectScreen. |
ACS Chem Biol 11: 1537-43 (2016)
Article DOI: 10.1021/acschembio.6b00250
BindingDB Entry DOI: 10.7270/Q29K491Z |
More data for this
Ligand-Target Pair | |
Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human)) | BDBM185152
(STK16-IN-1)Show InChI InChI=1S/C16H10FN3O2/c17-12-3-2-10(7-13(12)21)20-14(22)4-1-9-8-19-16-11(15(9)20)5-6-18-16/h1-8,21H,(H,18,19) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 1.07E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences
| Assay Description
The enzymatic assay was performed using the LifeTechnology SelectScreen. |
ACS Chem Biol 11: 1537-43 (2016)
Article DOI: 10.1021/acschembio.6b00250
BindingDB Entry DOI: 10.7270/Q29K491Z |
More data for this
Ligand-Target Pair | |
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha
(Homo sapiens (Human)) | BDBM185152
(STK16-IN-1)Show InChI InChI=1S/C16H10FN3O2/c17-12-3-2-10(7-13(12)21)20-14(22)4-1-9-8-19-16-11(15(9)20)5-6-18-16/h1-8,21H,(H,18,19) | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 4.86E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences
| Assay Description
The enzymatic assay was performed using the LifeTechnology SelectScreen. |
ACS Chem Biol 11: 1537-43 (2016)
Article DOI: 10.1021/acschembio.6b00250
BindingDB Entry DOI: 10.7270/Q29K491Z |
More data for this
Ligand-Target Pair | |
Serine/threonine-protein kinase mTOR
(Homo sapiens (Human)) | BDBM185152
(STK16-IN-1)Show InChI InChI=1S/C16H10FN3O2/c17-12-3-2-10(7-13(12)21)20-14(22)4-1-9-8-19-16-11(15(9)20)5-6-18-16/h1-8,21H,(H,18,19) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 5.56E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences
| Assay Description
The enzymatic assay was performed using the LifeTechnology SelectScreen. |
ACS Chem Biol 11: 1537-43 (2016)
Article DOI: 10.1021/acschembio.6b00250
BindingDB Entry DOI: 10.7270/Q29K491Z |
More data for this
Ligand-Target Pair | |
Phosphatidylinositol 3-kinase catalytic subunit type 3
(Homo sapiens (Human)) | BDBM185152
(STK16-IN-1)Show InChI InChI=1S/C16H10FN3O2/c17-12-3-2-10(7-13(12)21)20-14(22)4-1-9-8-19-16-11(15(9)20)5-6-18-16/h1-8,21H,(H,18,19) | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 7.94E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences
| Assay Description
The enzymatic assay was performed using the LifeTechnology SelectScreen. |
ACS Chem Biol 11: 1537-43 (2016)
Article DOI: 10.1021/acschembio.6b00250
BindingDB Entry DOI: 10.7270/Q29K491Z |
More data for this
Ligand-Target Pair | |
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta
(Homo sapiens (Human)) | BDBM185152
(STK16-IN-1)Show InChI InChI=1S/C16H10FN3O2/c17-12-3-2-10(7-13(12)21)20-14(22)4-1-9-8-19-16-11(15(9)20)5-6-18-16/h1-8,21H,(H,18,19) | NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 9.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences
| Assay Description
The enzymatic assay was performed using the LifeTechnology SelectScreen. |
ACS Chem Biol 11: 1537-43 (2016)
Article DOI: 10.1021/acschembio.6b00250
BindingDB Entry DOI: 10.7270/Q29K491Z |
More data for this
Ligand-Target Pair | |
Phosphatidylinositol 4-kinase beta
(Homo sapiens (Human)) | BDBM185152
(STK16-IN-1)Show InChI InChI=1S/C16H10FN3O2/c17-12-3-2-10(7-13(12)21)20-14(22)4-1-9-8-19-16-11(15(9)20)5-6-18-16/h1-8,21H,(H,18,19) | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences
| Assay Description
The enzymatic assay was performed using the LifeTechnology SelectScreen. |
ACS Chem Biol 11: 1537-43 (2016)
Article DOI: 10.1021/acschembio.6b00250
BindingDB Entry DOI: 10.7270/Q29K491Z |
More data for this
Ligand-Target Pair | |
Phosphatidylinositol 4-kinase alpha
(Homo sapiens (Human)) | BDBM185152
(STK16-IN-1)Show InChI InChI=1S/C16H10FN3O2/c17-12-3-2-10(7-13(12)21)20-14(22)4-1-9-8-19-16-11(15(9)20)5-6-18-16/h1-8,21H,(H,18,19) | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences
| Assay Description
The enzymatic assay was performed using the LifeTechnology SelectScreen. |
ACS Chem Biol 11: 1537-43 (2016)
Article DOI: 10.1021/acschembio.6b00250
BindingDB Entry DOI: 10.7270/Q29K491Z |
More data for this
Ligand-Target Pair | |
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