Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405943 (CHEMBL176596) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 96 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405931 (CHEMBL367753) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405937 (CHEMBL173782) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405942 (CHEMBL175345) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 630 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405939 (CHEMBL175307) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50018055 (7-Amino-heptan-2-one | CHEMBL176843) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents | PubMed | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405932 (CHEMBL176530) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405935 (CHEMBL177305) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405928 (CHEMBL174669) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 7.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405940 (CHEMBL177890) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405930 (CHEMBL174887) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 1.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405934 (CHEMBL176764) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405929 (CHEMBL436093) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.76E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405941 (CHEMBL177777) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405938 (CHEMBL81241) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | PubMed | 8.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405933 (CHEMBL176800) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem | PubMed | 1.37E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisomal N(1)-acetyl-spermine/spermidine oxidase (Homo sapiens (Human)) | BDBM50405936 (CHEMBL177217) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 2.90E+7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of the Pacific Curated by ChEMBL | Assay Description Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver. | J Med Chem 32: 984-9 (1989) BindingDB Entry DOI: 10.7270/Q23777PG | |||||||||||
More data for this Ligand-Target Pair |