Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
RAC-alpha serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50182752 (CHEMBL3818018) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.13E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Milano-Bicocca Curated by ChEMBL | Assay Description Inhibition of human Akt1 PH domain using AKTide-2T as substrate by ELISA | Bioorg Med Chem 24: 3396-405 (2016) Article DOI: 10.1016/j.bmc.2016.05.031 BindingDB Entry DOI: 10.7270/Q2SF2Z2G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RAC-alpha serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50431630 (KRX-0401 | PERIFOSINE) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.34E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Milano-Bicocca Curated by ChEMBL | Assay Description Inhibition of human Akt1 PH domain using AKTide-2T as substrate by ELISA | Bioorg Med Chem 24: 3396-405 (2016) Article DOI: 10.1016/j.bmc.2016.05.031 BindingDB Entry DOI: 10.7270/Q2SF2Z2G | |||||||||||
More data for this Ligand-Target Pair |