Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human)) | BDBM16673 (4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | 7.4 | n/a |
Bharati Vidyapeeth's College of Pharmacy | Assay Description The inhibition was carried out in 96-well polystyrene round bottomed plates. These plates were precoated with 100 ul per well of 50 ug per ml poly(... | Bioorg Chem 67: 139-47 (2016) Article DOI: 10.1016/j.bioorg.2016.06.006 BindingDB Entry DOI: 10.7270/Q2GH9GR6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human)) | BDBM192706 (2-[4-(2,4-Dioxothiazolidin-5-ylidenemethyl)phenoxy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | 7.4 | n/a |
Bharati Vidyapeeth's College of Pharmacy | Assay Description The inhibition was carried out in 96-well polystyrene round bottomed plates. These plates were precoated with 100 ul per well of 50 ug per ml poly(... | Bioorg Chem 67: 139-47 (2016) Article DOI: 10.1016/j.bioorg.2016.06.006 BindingDB Entry DOI: 10.7270/Q2GH9GR6 | |||||||||||
More data for this Ligand-Target Pair |