Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prostaglandin G/H synthase 1 (Ovis aries (Sheep)) | BDBM13065 (5-(4-chlorophenyl)-1-(4-methoxyphenyl)-3-(trifluor...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 66 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 2 (Homo sapiens (Human)) | BDBM50029600 (5-Bromo-2-(4-fluoro-phenyl)-3-(4-methanesulfonyl-p...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 2 (Homo sapiens (Human)) | BDBM202550 (N-{4-[(1Z)-1-(hydroxyimino)ethyl]phenyl}-2-{[5-(3,...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 750 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 1 (Ovis aries (Sheep)) | BDBM202549 (N-{4-[(1Z)-1-(hydroxyimino)ethyl]phenyl}-2-{[5-(4-...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 980 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 1 (Ovis aries (Sheep)) | BDBM202547 (N-(4-acetylphenyl)-2-[(5-phenyl-1,3,4-oxadiazol-2-...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 1 (Ovis aries (Sheep)) | BDBM202550 (N-{4-[(1Z)-1-(hydroxyimino)ethyl]phenyl}-2-{[5-(3,...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.12E+3 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 2 (Homo sapiens (Human)) | BDBM202549 (N-{4-[(1Z)-1-(hydroxyimino)ethyl]phenyl}-2-{[5-(4-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 2 (Homo sapiens (Human)) | BDBM202547 (N-(4-acetylphenyl)-2-[(5-phenyl-1,3,4-oxadiazol-2-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.10E+3 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 2 (Homo sapiens (Human)) | BDBM202548 (N-(4-acetylphenyl)-2-{[5-(4-chlorophenyl)-1,3,4-ox...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.90E+3 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 1 (Ovis aries (Sheep)) | BDBM202548 (N-(4-acetylphenyl)-2-{[5-(4-chlorophenyl)-1,3,4-ox...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.03E+4 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 1 (Ovis aries (Sheep)) | BDBM202551 (N-(4-acetylphenyl)-2-[(5-{1-[4-(2-methylpropyl)phe...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.03E+4 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 2 (Homo sapiens (Human)) | BDBM202551 (N-(4-acetylphenyl)-2-[(5-{1-[4-(2-methylpropyl)phe...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.05E+4 | n/a | n/a | n/a | n/a | 8.0 | 25 |
Minia University | Assay Description COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz... | Bioorg Chem 69: 48-63 (2016) Article DOI: 10.1016/j.bioorg.2016.09.005 BindingDB Entry DOI: 10.7270/Q21J98KS | |||||||||||
More data for this Ligand-Target Pair |