Affinity Data by PubMed id=2883317

PubMed code 2883317

Found 6 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Beta-1/Beta-2/Beta-3 adrenergic receptor (Rattus norvegicus (Rat))	BDBM25761 (Anapriline \| Avlocardyl \| CHEMBL27 \| PROPANOLOL(-)...) Show SMILES CC(C)NCC(O)COc1cccc2ccccc12 Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars	PubMed	6.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Evaluated for beta-receptor affinity determined in rat brain membrane fraction with [3H]- dihydroalprenolol				J Med Chem 30: 788-92 (1987) BindingDB Entry DOI: 10.7270/Q2FT8P8T
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Beta-1/Beta-2/Beta-3 adrenergic receptor (Rattus norvegicus (Rat))	BDBM50226764 (CHEMBL1203802) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Evaluated for beta-receptor affinity, determined in rat brain membrane fraction with [3H]- dihydroalprenolol				J Med Chem 30: 788-92 (1987) BindingDB Entry DOI: 10.7270/Q2FT8P8T
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Beta-1/Beta-2/Beta-3 adrenergic receptor (Rattus norvegicus (Rat))	BDBM50226766 (CHEMBL354278) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Evaluated for beta-receptor affinity, determined in rat brain membrane fraction with [3H]- dihydroalprenolol				J Med Chem 30: 788-92 (1987) BindingDB Entry DOI: 10.7270/Q2FT8P8T
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Beta-1/Beta-2/Beta-3 adrenergic receptor (Rattus norvegicus (Rat))	BDBM50226763 (CHEMBL1203804) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Evaluated for beta-receptor affinity determined in rat brain membrane fraction with [3H]- dihydroalprenolol				J Med Chem 30: 788-92 (1987) BindingDB Entry DOI: 10.7270/Q2FT8P8T
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Beta-1/Beta-2/Beta-3 adrenergic receptor (Rattus norvegicus (Rat))	BDBM50226762 (CHEMBL423629) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Evaluated for beta-receptor affinity, determined in rat brain membrane fraction with [3H]- dihydroalprenolol				J Med Chem 30: 788-92 (1987) BindingDB Entry DOI: 10.7270/Q2FT8P8T
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Beta-1/Beta-2/Beta-3 adrenergic receptor (Rattus norvegicus (Rat))	BDBM50226765 (CHEMBL58430) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Evaluated for beta-receptor affinity, determined in rat brain membrane fraction with [3H]- dihydroalprenolol				J Med Chem 30: 788-92 (1987) BindingDB Entry DOI: 10.7270/Q2FT8P8T
TBA Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%