Affinity Data by BDB articleid=50029418

Articleid 50029418

Found 3 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Type-1 angiotensin II receptor (Homo sapiens (Human))	BDBM50284297 (4-(2-Butyl-5-{[(R)-1-carboxy-2-(1H-indol-3-yl)-eth...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	2.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Tested for inhibition of Angiotensin II specific binding to Angiotensin II receptor, type 1 in the recombinant human AT-1 receptor expressed in LhAT-...				Bioorg Med Chem Lett 5: 19-24 (1995) Article DOI: 10.1016/0960-894X(94)00456-P BindingDB Entry DOI: 10.7270/Q2GF0TF6
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Type-1 angiotensin II receptor (Homo sapiens (Human))	BDBM50284298 (4-(2-Butyl-5-{[(S)-1-carboxy-2-(1H-indol-3-yl)-eth...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	48.3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Tested for inhibition of Angiotensin II specific binding to Angiotensin II receptor, type 1 in the recombinant human AT-1 receptor expressed in LhAT-...				Bioorg Med Chem Lett 5: 19-24 (1995) Article DOI: 10.1016/0960-894X(94)00456-P BindingDB Entry DOI: 10.7270/Q2GF0TF6
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Type-1 angiotensin II receptor (Homo sapiens (Human))	BDBM50284295 (4-{2-Butyl-5-[(carboxymethyl-amino)-methyl]-imidaz...) Show SMILES CCCCc1ncc(CNCC(O)=O)n1Cc1ccc(cc1)C(O)=O Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	298	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Tested for inhibition of Angiotensin II specific binding to Angiotensin II receptor, type 1 in the recombinant human AT-1 receptor expressed in LhAT-...				Bioorg Med Chem Lett 5: 19-24 (1995) Article DOI: 10.1016/0960-894X(94)00456-P BindingDB Entry DOI: 10.7270/Q2GF0TF6
TBA Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%