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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50280478 (BB-823 | CHEMBL157078 | N-((S)-1-Ethoxymethyl-3-me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet  | CHEMBL PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | 0.0150 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonistic activity for inhibition of [3H]PAF receptor binding to washed human platelet membranes. | Bioorg Med Chem Lett 2: 597-602 (1992) Article DOI: 10.1016/S0960-894X(01)81205-1 BindingDB Entry DOI: 10.7270/Q2CF9QK7 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50280480 (CHEMBL156461 | YM-461 | [4-(3-Phenyl-propyl)-piper...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonistic activity for inhibition of [3H]PAF receptor binding to washed human platelet membranes. | Bioorg Med Chem Lett 2: 597-602 (1992) Article DOI: 10.1016/S0960-894X(01)81205-1 BindingDB Entry DOI: 10.7270/Q2CF9QK7 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50280479 ((R)-3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazole-7-car...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonistic activity for inhibition of [3H]PAF receptor binding to washed human platelet membranes. | Bioorg Med Chem Lett 2: 597-602 (1992) Article DOI: 10.1016/S0960-894X(01)81205-1 BindingDB Entry DOI: 10.7270/Q2CF9QK7 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50004633 ((S)-4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-im...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonistic activity for inhibition of [3H]PAF receptor binding to washed human platelet membranes. | Bioorg Med Chem Lett 2: 597-602 (1992) Article DOI: 10.1016/S0960-894X(01)81205-1 BindingDB Entry DOI: 10.7270/Q2CF9QK7 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011671 ((2E,4E)-5-(4-Methoxy-phenyl)-deca-2,4-dienoic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonistic activity for inhibition of [3H]PAF receptor binding to washed human platelet membranes. | Bioorg Med Chem Lett 2: 597-602 (1992) Article DOI: 10.1016/S0960-894X(01)81205-1 BindingDB Entry DOI: 10.7270/Q2CF9QK7 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50000714 (3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonistic activity for inhibition of [3H]PAF receptor binding to washed human platelet membranes. | Bioorg Med Chem Lett 2: 597-602 (1992) Article DOI: 10.1016/S0960-894X(01)81205-1 BindingDB Entry DOI: 10.7270/Q2CF9QK7 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50280482 (BB-182 | CHEMBL418608 | N-Cyclohexyl-N-methyl-4-(2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonistic activity for inhibition of [3H]PAF receptor binding to washed human platelet membranes. | Bioorg Med Chem Lett 2: 597-602 (1992) Article DOI: 10.1016/S0960-894X(01)81205-1 BindingDB Entry DOI: 10.7270/Q2CF9QK7 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50280477 (BB-350 | CHEMBL345902 | N-Cyclohexyl-N-methyl-4-(2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonistic activity for inhibition of [3H]PAF receptor binding to washed human platelet membranes. | Bioorg Med Chem Lett 2: 597-602 (1992) Article DOI: 10.1016/S0960-894X(01)81205-1 BindingDB Entry DOI: 10.7270/Q2CF9QK7 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
