Affinity Data by BDB articleid=50040998

Articleid 50040998

Found 3 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Histamine H2 receptor (RAT)	BDBM22881 (5-(2-aminoethyl)-4-methyl-1,3-thiazol-2-amine \| Am...) Show SMILES Cc1nc(N)sc1CCN Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article	n/a	n/a	n/a	1.15E+4	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligand				Bioorg Med Chem Lett 4: 1913-1916 (1994) Article DOI: 10.1016/S0960-894X(01)80533-3 BindingDB Entry DOI: 10.7270/Q2TD9ZHX
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Histamine H2 receptor (RAT)	BDBM22882 (2-amino-5(2-aminoethyl)-4-methyl-1,3-selenazole \| ...) Show SMILES Cc1nc(N)[se]c1CCN Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	n/a	9.77E+3	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligand				Bioorg Med Chem Lett 4: 1913-1916 (1994) Article DOI: 10.1016/S0960-894X(01)80533-3 BindingDB Entry DOI: 10.7270/Q2TD9ZHX
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Histamine H2 receptor (RAT)	BDBM7966 (2-(1H-imidazol-4-yl)ethan-1-amine \| CHEMBL544208 \|...) Show SMILES NCCc1cnc[nH]1 Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars	Article	n/a	n/a	n/a	1.17E+5	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligand				Bioorg Med Chem Lett 4: 1913-1916 (1994) Article DOI: 10.1016/S0960-894X(01)80533-3 BindingDB Entry DOI: 10.7270/Q2TD9ZHX
TBA Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%