Affinity Data by PubMed id=7658433

PubMed code 7658433

Found 27 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig))	BDBM50033139 (CHEMBL2370495 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	0.240	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig))	BDBM50453783 (CHEMBL2311023) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	0.550	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig))	BDBM50033143 (CHEMBL216640 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	0.580	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig))	BDBM50453785 (CHEMBL2311025) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	0.610	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50453785 (CHEMBL2311025) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	0.640	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGO				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig))	BDBM50453782 (CHEMBL2370497) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	0.900	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50033142 (CHEMBL2370496 \| H-Tyr-Gly-Gly-Phe-Leu-Lys-Arg-Il...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	4	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGO				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig))	BDBM50033142 (CHEMBL2370496 \| H-Tyr-Gly-Gly-Phe-Leu-Lys-Arg-Il...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	4	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50033139 (CHEMBL2370495 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	5.20	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGO				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig))	BDBM50453784 (CHEMBL2311024) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	8	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50453782 (CHEMBL2370497) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	9	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGO				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50033141 (CHEMBL2370494 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys*-Ile...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	9.20	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGO				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50033143 (CHEMBL216640 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	9.90	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGO				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50453783 (CHEMBL2311023) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	12	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGO				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50033142 (CHEMBL2370496 \| H-Tyr-Gly-Gly-Phe-Leu-Lys-Arg-Il...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	13	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalin				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50033141 (CHEMBL2370494 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys*-Ile...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	17	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalin				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig))	BDBM50033141 (CHEMBL2370494 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys*-Ile...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	17	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50033139 (CHEMBL2370495 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	18	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalin				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50453783 (CHEMBL2311023) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	24	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalin				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50033143 (CHEMBL216640 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	26	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalin				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50453785 (CHEMBL2311025) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	32	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalin				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50453782 (CHEMBL2370497) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	53	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalin				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50453784 (CHEMBL2311024) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	96	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGO				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50453784 (CHEMBL2311024) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	198	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalin				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (GUINEA PIG)	BDBM50033137 (CHEMBL2311022 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	1.04E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGO				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig))	BDBM50033137 (CHEMBL2311022 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	7.99E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair
Delta-type opioid receptor (Homo sapiens (Human))	BDBM50033137 (CHEMBL2311022 \| H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	8.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Arizona Curated by ChEMBL					Assay Description Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalin				J Med Chem 38: 3462-8 (1995) BindingDB Entry DOI: 10.7270/Q2QZ291Q
University of Arizona Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%