Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Delta-type opioid receptor (MOUSE) | BDBM50041669 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferens | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50041669 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50041663 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 42 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50453339 (CHEMBL2372412) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 66 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (MOUSE) | BDBM50453339 (CHEMBL2372412) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 85 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferens | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (MOUSE) | BDBM50041663 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferens | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (MOUSE) | BDBM50001683 (13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 570 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferens | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50001683 (13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (MOUSE) | BDBM50041666 (2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 760 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferens | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50041666 (2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 760 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50453339 (CHEMBL2372412) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexus | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50001683 (13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexus | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50041669 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50453339 (CHEMBL2372412) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50041663 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >2.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (MOUSE) | BDBM50041668 (2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferens | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50041668 (2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50041668 (2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexus | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50041665 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50041665 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (MOUSE) | BDBM50041665 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferens | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50041665 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexus | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50001683 (13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50041663 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexus | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50041668 (2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50041666 (2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP binding | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50041669 (2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexus | J Med Chem 37: 1572-7 (1994) BindingDB Entry DOI: 10.7270/Q2DR2W47 | |||||||||||
More data for this Ligand-Target Pair |