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PubMed code 9873693

Compile data set for download or QSAR
Found 24 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Mu-type opioid receptor


(GUINEA PIG)		BDBM60212
PNG
((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Show SMILES Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)CC[C@@]35O
Show InChI InChI=1S/C20H23NO4/c22-13-4-3-12-9-15-20(24)6-5-14(23)18-19(20,16(12)17(13)25-18)7-8-21(15)10-11-1-2-11/h3-4,11,15,18,22,24H,1-2,5-10H2/t15-,18+,19+,20-/m1/s1
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 0.560n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined as ability to displace [3H]-U-69, radioligand from Opioid receptor kappa 1

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM60212
PNG
((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Show SMILES Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)CC[C@@]35O
Show InChI InChI=1S/C20H23NO4/c22-13-4-3-12-9-15-20(24)6-5-14(23)18-19(20,16(12)17(13)25-18)7-8-21(15)10-11-1-2-11/h3-4,11,15,18,22,24H,1-2,5-10H2/t15-,18+,19+,20-/m1/s1
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 0.930n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Compound was tested for the inhibition of [35S]-GTP-gammaS, binding in Guinea pig Caudate stimulated by the opioid receptor agonist Mu-DAMGO

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(Rattus norvegicus (rat))		BDBM60212
PNG
((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Show SMILES Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)CC[C@@]35O
Show InChI InChI=1S/C20H23NO4/c22-13-4-3-12-9-15-20(24)6-5-14(23)18-19(20,16(12)17(13)25-18)7-8-21(15)10-11-1-2-11/h3-4,11,15,18,22,24H,1-2,5-10H2/t15-,18+,19+,20-/m1/s1
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 1.40n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined as ability to displace [3H]-DAMGO radioligand from Mu opioid receptor

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50045767
PNG
((+)-N-phenethyl trans-3(R),4(R)-dimethyl-4-(3-hydr...)
Show SMILES C[C@H]1CN(CCc2ccccc2)CC[C@@]1(C)c1cccc(O)c1
Show InChI InChI=1S/C21H27NO/c1-17-16-22(13-11-18-7-4-3-5-8-18)14-12-21(17,2)19-9-6-10-20(23)15-19/h3-10,15,17,23H,11-14,16H2,1-2H3/t17-,21+/m0/s1
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 1.5n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined against Mu opioid receptor using [3H]-Naltrexone as radioligand

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM60212
PNG
((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Show SMILES Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)CC[C@@]35O
Show InChI InChI=1S/C20H23NO4/c22-13-4-3-12-9-15-20(24)6-5-14(23)18-19(20,16(12)17(13)25-18)7-8-21(15)10-11-1-2-11/h3-4,11,15,18,22,24H,1-2,5-10H2/t15-,18+,19+,20-/m1/s1
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 2.10n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined against Mu opioid receptor using [3H]naltrexone as radioligand

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM60212
PNG
((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Show SMILES Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)CC[C@@]35O
Show InChI InChI=1S/C20H23NO4/c22-13-4-3-12-9-15-20(24)6-5-14(23)18-19(20,16(12)17(13)25-18)7-8-21(15)10-11-1-2-11/h3-4,11,15,18,22,24H,1-2,5-10H2/t15-,18+,19+,20-/m1/s1
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 3.90n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined against Opioid receptor kappa 1
using [3H]-Ethylketocyclazocine as radioligand

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM60212
PNG
((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Show SMILES Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)CC[C@@]35O
Show InChI InChI=1S/C20H23NO4/c22-13-4-3-12-9-15-20(24)6-5-14(23)18-19(20,16(12)17(13)25-18)7-8-21(15)10-11-1-2-11/h3-4,11,15,18,22,24H,1-2,5-10H2/t15-,18+,19+,20-/m1/s1
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 4.70n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Compound was tested for the inhibition of [35S]-GTP-gammaS, binding to Opioid receptor kappa 1

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50072452
PNG
(3-((4aS,10aS)-10a-Methyl-2-phenethyl-1,3,4,5,10,10...)
Show SMILES C[C@@]12CN(CCc3ccccc3)CC[C@@]1(Cc1ccccc1C2)c1cccc(O)c1
Show InChI InChI=1S/C28H31NO/c1-27-19-23-10-5-6-11-24(23)20-28(27,25-12-7-13-26(30)18-25)15-17-29(21-27)16-14-22-8-3-2-4-9-22/h2-13,18,30H,14-17,19-21H2,1H3/t27-,28-/m1/s1
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 6.60n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Compound was tested for the inhibition of [35S]-GTP-gammaS, binding Opioid receptor kappa 1

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50072452
PNG
(3-((4aS,10aS)-10a-Methyl-2-phenethyl-1,3,4,5,10,10...)
Show SMILES C[C@@]12CN(CCc3ccccc3)CC[C@@]1(Cc1ccccc1C2)c1cccc(O)c1
Show InChI InChI=1S/C28H31NO/c1-27-19-23-10-5-6-11-24(23)20-28(27,25-12-7-13-26(30)18-25)15-17-29(21-27)16-14-22-8-3-2-4-9-22/h2-13,18,30H,14-17,19-21H2,1H3/t27-,28-/m1/s1
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 9.80n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Compound was tested for the inhibition of [35S]-GTP-gammaS, binding to Opioid receptor kappa 1

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50072452
PNG
(3-((4aS,10aS)-10a-Methyl-2-phenethyl-1,3,4,5,10,10...)
Show SMILES C[C@@]12CN(CCc3ccccc3)CC[C@@]1(Cc1ccccc1C2)c1cccc(O)c1
Show InChI InChI=1S/C28H31NO/c1-27-19-23-10-5-6-11-24(23)20-28(27,25-12-7-13-26(30)18-25)15-17-29(21-27)16-14-22-8-3-2-4-9-22/h2-13,18,30H,14-17,19-21H2,1H3/t27-,28-/m1/s1
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 10n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Compound was tested for the inhibition of [35S]-GTP-gammaS, binding in Guinea pig Caudate stimulated by the opioid receptor agonist Mu-DAMGO

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(Rattus norvegicus (rat))		BDBM50072452
PNG
(3-((4aS,10aS)-10a-Methyl-2-phenethyl-1,3,4,5,10,10...)
Show SMILES C[C@@]12CN(CCc3ccccc3)CC[C@@]1(Cc1ccccc1C2)c1cccc(O)c1
Show InChI InChI=1S/C28H31NO/c1-27-19-23-10-5-6-11-24(23)20-28(27,25-12-7-13-26(30)18-25)15-17-29(21-27)16-14-22-8-3-2-4-9-22/h2-13,18,30H,14-17,19-21H2,1H3/t27-,28-/m1/s1
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 11n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined as ability to displace [3H]-DAMGO radioligand from Mu opioid receptor

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Homo sapiens (Human))		BDBM60212
PNG
((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Show SMILES Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)CC[C@@]35O
Show InChI InChI=1S/C20H23NO4/c22-13-4-3-12-9-15-20(24)6-5-14(23)18-19(20,16(12)17(13)25-18)7-8-21(15)10-11-1-2-11/h3-4,11,15,18,22,24H,1-2,5-10H2/t15-,18+,19+,20-/m1/s1
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 19n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Compound was tested for the inhibition of [35S]-GTP-gammaS, binding in Guinea pig Caudate stimulated by the Opioid receptor delta 1 agonist Delta-SNC...

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50045767
PNG
((+)-N-phenethyl trans-3(R),4(R)-dimethyl-4-(3-hydr...)
Show SMILES C[C@H]1CN(CCc2ccccc2)CC[C@@]1(C)c1cccc(O)c1
Show InChI InChI=1S/C21H27NO/c1-17-16-22(13-11-18-7-4-3-5-8-18)14-12-21(17,2)19-9-6-10-20(23)15-19/h3-10,15,17,23H,11-14,16H2,1-2H3/t17-,21+/m0/s1
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 52n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined against Opioid receptor kappa 1
using [3H]-Ethylketocyclazocine as radioligand

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50072453
PNG
(3-((4aS,10aS)-2,10a-Dimethyl-1,3,4,5,10,10a-hexahy...)
Show SMILES CN1CC[C@@]2(Cc3ccccc3C[C@]2(C)C1)c1cccc(O)c1
Show InChI InChI=1S/C21H25NO/c1-20-13-16-6-3-4-7-17(16)14-21(20,10-11-22(2)15-20)18-8-5-9-19(23)12-18/h3-9,12,23H,10-11,13-15H2,1-2H3/t20-,21-/m1/s1
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 53n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined as ability to displace [3H]-U-69, radioligand from Opioid receptor kappa 1

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50045772
PNG
(3-((3R,4R)-1,3,4-Trimethyl-piperidin-4-yl)-phenol ...)
Show SMILES C[C@H]1CN(C)CC[C@@]1(C)c1cccc(O)c1
Show InChI InChI=1S/C14H21NO/c1-11-10-15(3)8-7-14(11,2)12-5-4-6-13(16)9-12/h4-6,9,11,16H,7-8,10H2,1-3H3/t11-,14+/m0/s1
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 80n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined against Mu opioid receptor using [3H]-Naltrexone as radioligand

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Rattus norvegicus (rat))		BDBM60212
PNG
((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Show SMILES Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)CC[C@@]35O
Show InChI InChI=1S/C20H23NO4/c22-13-4-3-12-9-15-20(24)6-5-14(23)18-19(20,16(12)17(13)25-18)7-8-21(15)10-11-1-2-11/h3-4,11,15,18,22,24H,1-2,5-10H2/t15-,18+,19+,20-/m1/s1
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 95n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined as ability to displace [3H]-DADLE radioligand from Opioid receptor delta 1

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(GUINEA PIG)		BDBM50072453
PNG
(3-((4aS,10aS)-2,10a-Dimethyl-1,3,4,5,10,10a-hexahy...)
Show SMILES CN1CC[C@@]2(Cc3ccccc3C[C@]2(C)C1)c1cccc(O)c1
Show InChI InChI=1S/C21H25NO/c1-20-13-16-6-3-4-7-17(16)14-21(20,10-11-22(2)15-20)18-8-5-9-19(23)12-18/h3-9,12,23H,10-11,13-15H2,1-2H3/t20-,21-/m1/s1
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 119n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Compound was tested for the inhibition of [35S]-GTP-gammaS, binding in Guinea pig Caudate stimulated by the opioid receptor agonist Mu-DAMGO

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50072453
PNG
(3-((4aS,10aS)-2,10a-Dimethyl-1,3,4,5,10,10a-hexahy...)
Show SMILES CN1CC[C@@]2(Cc3ccccc3C[C@]2(C)C1)c1cccc(O)c1
Show InChI InChI=1S/C21H25NO/c1-20-13-16-6-3-4-7-17(16)14-21(20,10-11-22(2)15-20)18-8-5-9-19(23)12-18/h3-9,12,23H,10-11,13-15H2,1-2H3/t20-,21-/m1/s1
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 166n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined as ability to displace [3H]-U-69, radioligand from Opioid receptor kappa 1

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Homo sapiens (Human))		BDBM50072452
PNG
(3-((4aS,10aS)-10a-Methyl-2-phenethyl-1,3,4,5,10,10...)
Show SMILES C[C@@]12CN(CCc3ccccc3)CC[C@@]1(Cc1ccccc1C2)c1cccc(O)c1
Show InChI InChI=1S/C28H31NO/c1-27-19-23-10-5-6-11-24(23)20-28(27,25-12-7-13-26(30)18-25)15-17-29(21-27)16-14-22-8-3-2-4-9-22/h2-13,18,30H,14-17,19-21H2,1H3/t27-,28-/m1/s1
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 184n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Compound was tested for the inhibition of [35S]-GTP-gammaS, binding in Guinea pig Caudate stimulated by the Opioid receptor delta 1 agonist Delta-SNC...

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Homo sapiens (Human))		BDBM50072453
PNG
(3-((4aS,10aS)-2,10a-Dimethyl-1,3,4,5,10,10a-hexahy...)
Show SMILES CN1CC[C@@]2(Cc3ccccc3C[C@]2(C)C1)c1cccc(O)c1
Show InChI InChI=1S/C21H25NO/c1-20-13-16-6-3-4-7-17(16)14-21(20,10-11-22(2)15-20)18-8-5-9-19(23)12-18/h3-9,12,23H,10-11,13-15H2,1-2H3/t20-,21-/m1/s1
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 222n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Compound was tested for the inhibition of [35S]-GTP-gammaS, binding in Guinea pig Caudate stimulated by the Opioid receptor delta 1 agonist Delta-SNC...

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Mu-type opioid receptor


(Rattus norvegicus (rat))		BDBM50072453
PNG
(3-((4aS,10aS)-2,10a-Dimethyl-1,3,4,5,10,10a-hexahy...)
Show SMILES CN1CC[C@@]2(Cc3ccccc3C[C@]2(C)C1)c1cccc(O)c1
Show InChI InChI=1S/C21H25NO/c1-20-13-16-6-3-4-7-17(16)14-21(20,10-11-22(2)15-20)18-8-5-9-19(23)12-18/h3-9,12,23H,10-11,13-15H2,1-2H3/t20-,21-/m1/s1
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 297n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined as ability to displace [3H]-DAMGO radioligand from Mu opioid receptor

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Kappa-type opioid receptor


(Cavia porcellus (domestic guinea pig))		BDBM50045772
PNG
(3-((3R,4R)-1,3,4-Trimethyl-piperidin-4-yl)-phenol ...)
Show SMILES C[C@H]1CN(C)CC[C@@]1(C)c1cccc(O)c1
Show InChI InChI=1S/C14H21NO/c1-11-10-15(3)8-7-14(11,2)12-5-4-6-13(16)9-12/h4-6,9,11,16H,7-8,10H2,1-3H3/t11-,14+/m0/s1
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 833n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined against Opioid receptor kappa 1
using [3H]-Ethylketocyclazocine as radioligand

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Rattus norvegicus (rat))		BDBM50072452
PNG
(3-((4aS,10aS)-10a-Methyl-2-phenethyl-1,3,4,5,10,10...)
Show SMILES C[C@@]12CN(CCc3ccccc3)CC[C@@]1(Cc1ccccc1C2)c1cccc(O)c1
Show InChI InChI=1S/C28H31NO/c1-27-19-23-10-5-6-11-24(23)20-28(27,25-12-7-13-26(30)18-25)15-17-29(21-27)16-14-22-8-3-2-4-9-22/h2-13,18,30H,14-17,19-21H2,1H3/t27-,28-/m1/s1
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 1.27E+3n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined as ability to displace [3H]-DADLE radioligand from Opioid receptor delta 1

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
Delta-type opioid receptor


(Rattus norvegicus (rat))		BDBM50072453
PNG
(3-((4aS,10aS)-2,10a-Dimethyl-1,3,4,5,10,10a-hexahy...)
Show SMILES CN1CC[C@@]2(Cc3ccccc3C[C@]2(C)C1)c1cccc(O)c1
Show InChI InChI=1S/C21H25NO/c1-20-13-16-6-3-4-7-17(16)14-21(20,10-11-22(2)15-20)18-8-5-9-19(23)12-18/h3-9,12,23H,10-11,13-15H2,1-2H3/t20-,21-/m1/s1
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>5.71E+3n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity was determined as ability to displace [3H]-DADLE radioligand from Opioid receptor delta 1

Bioorg Med Chem Lett 8: 3149-52 (1999)


BindingDB Entry DOI: 10.7270/Q2S75FGQ
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%