Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Beta-lactamase (Pseudomonas aeruginosa (PAO1)) | BDBM212440 (US8772490, H) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 650 | n/a | n/a | n/a | n/a | 7.0 | 30 |
Meiji Seika Pharma Co., Ltd. US Patent | Assay Description For the measurement of β-lactamase inhibitory activity, 100 uM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% DMSO, ... | US Patent US8772490 (2014) BindingDB Entry DOI: 10.7270/Q2NK3CWQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-lactamase (Pseudomonas aeruginosa (PAO1)) | BDBM159600 (US8772490, Example 23 | US9035062, 23) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 650 | n/a | n/a | n/a | n/a | 7.0 | 30 |
Meiji Seika Pharma Co., Ltd. US Patent | Assay Description For the measurement of β-lactamase inhibitory activity, 100 uM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% DMSO, ... | US Patent US8772490 (2014) BindingDB Entry DOI: 10.7270/Q2NK3CWQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-lactamase (Pseudomonas aeruginosa (PAO1)) | BDBM212441 (US8772490, TAZ) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 950 | n/a | n/a | n/a | n/a | 7.0 | 30 |
Meiji Seika Pharma Co., Ltd. US Patent | Assay Description For the measurement of β-lactamase inhibitory activity, 100 uM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% DMSO, ... | US Patent US8772490 (2014) BindingDB Entry DOI: 10.7270/Q2NK3CWQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-lactamase (Pseudomonas aeruginosa (PAO1)) | BDBM159601 (US8772490, Example 24 | US9035062, 24) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | 7.0 | 30 |
Meiji Seika Pharma Co., Ltd. US Patent | Assay Description For the measurement of β-lactamase inhibitory activity, 100 uM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% DMSO, ... | US Patent US8772490 (2014) BindingDB Entry DOI: 10.7270/Q2NK3CWQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-lactamase (Pseudomonas aeruginosa (PAO1)) | BDBM159601 (US8772490, Example 24 | US9035062, 24) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | 7.0 | 30 |
Meiji Seika Pharma Co., Ltd. US Patent | Assay Description For the measurement of β-lactamase inhibitory activity, 100 uM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% DMSO, ... | US Patent US8772490 (2014) BindingDB Entry DOI: 10.7270/Q2NK3CWQ | |||||||||||
More data for this Ligand-Target Pair |