Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Short transient receptor potential channel 4 (Mus musculus) | BDBM77625 (6-ethyl-4-methyl-2-(1-pyrrolidinyl)quinoline;2,2,2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 2.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM72595 (2-(1-azepanyl)-7-methoxy-4-methylquinoline;oxalic ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | PCBioAssay | n/a | n/a | 2.38E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77617 (4-methyl-2-(1-piperidinyl)quinoline | 4-methyl-2-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 2.63E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77618 (4-methyl-2-(4-methyl-1-piperidinyl)quinoline;2,2,2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 3.14E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77620 (4-methyl-2-(1-pyrrolidinyl)quinoline;2,2,2-trifluo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 3.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77624 (4,6-dimethyl-2-(1-pyrrolidinyl)quinoline;2,2,2-tri...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 3.71E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77621 (4-methyl-2-[(2S)-2-methyl-1-pyrrolidinyl]quinoline...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 4.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77614 ((4-Fluoro-benzyl)-[5-(4-fluoro-phenyl)-1-methyl-1H...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 4.28E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77616 (4-chloranyl-N'-cyclohexyl-benzenecarboximidamide;h...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | PCBioAssay | n/a | n/a | 4.56E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77623 (4,6-dimethyl-2-(1-piperidinyl)quinoline;2,2,2-trif...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 5.49E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77626 (6-fluoranyl-4-methyl-2-piperidin-1-yl-quinoline;2,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 6.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77622 (4-methyl-2-(4-pyridin-4-yl-1-piperazinyl)quinoline...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 8.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77615 (2-phenyl-N-(2-phenylsulfanylphenyl)acetamide | 2-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 3.87E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Short transient receptor potential channel 4 (Mus musculus) | BDBM77619 (4-(4-methyl-2-quinolinyl)morpholine;2,2,2-trifluor...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 1.40E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Johns Hopkins Ion Channel Center Curated by PubChem BioAssay | Assay Description Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2JS9NWF | |||||||||||
More data for this Ligand-Target Pair |