Reaction Details |
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Target | Casein kinase II subunit alpha |
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Ligand | BDBM8061 |
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Substrate/Competitor | CK2 Peptide Substrate |
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Meas. Tech. | CDK Inhibition Assay |
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Temperature | 303.15±n/a K |
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Ki | >1000±n/a nM |
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Comments | extracted |
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Citation | Wang, S; Wood, G; Meades, C; Griffiths, G; Midgley, C; McNae, I; McInnes, C; Anderson, S; Jackson, W; Mezna, M; Yuill, R; Walkinshaw, M; Fischer, PM Synthesis and biological activity of 2-anilino-4-(1H-pyrrol-3-yl) pyrimidine CDK inhibitors. Bioorg Med Chem Lett14:4237-40 (2004) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Casein kinase II subunit alpha |
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Name: | Casein kinase II subunit alpha |
Synonyms: | CK II | CK2 | CK2- alpha | CK2A1 | CSK21_HUMAN | CSNK2A1 | Casein kinase 2 | Casein kinase II (CK2) | Casein kinase II alpha/beta | Casein kinase II subunit alpha (CK2 alpha) | Casein kinase II subunit alpha (CK2A1) | Casein kinase II subunit alpha (CK2a I174A) | Casein kinase II subunit alpha (CK2a V66A) | Casein kinase II subunit alpha (CK2a dm V66I174AA) | Casein kinase II subunit alpha (CK2a) |
Type: | Enzyme |
Mol. Mass.: | 45151.12 |
Organism: | Homo sapiens (Human) |
Description: | P68400 |
Residue: | 391 |
Sequence: | MSGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINIT
NNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTD
FKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAE
FYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYD
QLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDF
LDKLLRYDHQSRLTAREAMEHPYFYTVVKDQARMGSSSMPGGSTPVSSANMMSGISSVPT
PSPLGPLAGSPVIAAANPLGMPVPAAAGAQQ
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BDBM8061 |
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CK2 Peptide Substrate |
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Name: | CK2 Peptide Substrate |
Synonyms: | n/a |
Type: | Peptide |
Mol. Mass.: | 1261.15 |
Organism: | n/a |
Description: | n/a |
Residue: | 10 |
Sequence: | |