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TargetPCAF (aa 719-832)
LigandBDBM311486
Substrate/Competitorn/a
Meas. Tech.PCAF AlphaLisa Binding Assay
IC50 19.0±n/a nM
Citation Albrecht BKCote ACrawford TDuplessis MGood ACLeBlanc YMagnuson SNasveschuk CGPastor RRomero AFTaylor AM Therapeutic compounds and uses thereof US Patent  US10155764 Publication Date 12/18/2018
More Info.:Get all data from this article,  Assay Method
 
PCAF (aa 719-832)
Name:PCAF (aa 719-832)
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:13536.05
Organism:Homo sapiens (Human)
Description:n/a
Residue:113
Sequence:
KEPRDPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKN
RYYVSKKLFMADLQRVFTNCKEYNPPESEYYKCANILEKFFFSKIKEAGLIDK
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM311486
n/a
NameBDBM311486
Synonyms:CHEM-US-00192 | US10155764, Example 65B
TypeSmall organic molecule
Emp. Form.C19H23N5O
Mol. Mass.337.4188
SMILESC[C@@H](Nc1nn(C)c(=O)c2cccnc12)[C@H](N(C)C)c1ccccc1 |r|
Structure
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