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Reaction Details
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TargetSigma intracellular receptor 2
LigandBDBM50374602
Substrate/Competitorn/a
Meas. Tech.Receptor Assay
Ki 1.49±0.18 nM
Citation McCurdy, CRMesangeau, CChin, FTJames, MLShen, BGambhir, S Highly selective sigma receptor radioligands US Patent US9604926 Publication Date 3/28/2017
More Info.:Get all data from this article,  Assay Method
 
Sigma intracellular receptor 2
Name:Sigma intracellular receptor 2
Synonyms:S2r | SGMR2_MOUSE | Sigma-2 receptor | Sigma2 receptor | Tmem97 | Transmembrane protein 97
Type:n/a
Mol. Mass.:20818.69
Organism:Mus musculus (Mouse)
Description:Q8VD00
Residue:176
Sequence:
MGALAARRCVEWLLGLYFVSHIPITLFIDLQAVLPPELYPQEFSNLLRWYSKEFKDPLMQ
EPPVWFKSFLLCELVFQLPFFPIAAYAFFKGSCRWIRIPAIIYAAHTITTLIPILYTLLF
EDFSKAVAFKGQRPESFRERLTLVGVYAPYLIIPLILLLFMLRNPYYKYEEKRKKK
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  Blast E-value cutoff:
BDBM50374602
n/a
NameBDBM50374602
Synonyms:CHEMBL272608 | US9604926, Compound SN-102 | US9724435, Compound SN-102
TypeSmall organic molecule
Emp. Form.C23H35N3OS
Mol. Mass.401.609
SMILESO=c1sc2ccccc2n1CCCCCCN1CCN(CC1)C1CCCCC1
Structure
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