| Reaction Details |
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 | Report a problem with these data |
| Target | Sigma intracellular receptor 2 |
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| Ligand | BDBM312203 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Receptor Assay |
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| Ki | 0.660±0.08 nM |
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| Citation |  McCurdy, CR; Mesangeau, C; Chin, FT; James, ML; Shen, B; Gambhir, S Highly selective sigma receptor radioligands US Patent US9604926 Publication Date 3/28/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| Sigma intracellular receptor 2 |
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| Name: | Sigma intracellular receptor 2 |
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| Synonyms: | S2r | SGMR2_MOUSE | Sigma-2 receptor | Sigma2 receptor | Tmem97 | Transmembrane protein 97 |
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| Type: | n/a |
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| Mol. Mass.: | 20818.69 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | Q8VD00 |
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| Residue: | 176 |
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| Sequence: | MGALAARRCVEWLLGLYFVSHIPITLFIDLQAVLPPELYPQEFSNLLRWYSKEFKDPLMQ
EPPVWFKSFLLCELVFQLPFFPIAAYAFFKGSCRWIRIPAIIYAAHTITTLIPILYTLLF
EDFSKAVAFKGQRPESFRERLTLVGVYAPYLIIPLILLLFMLRNPYYKYEEKRKKK
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| BDBM312203 |
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| n/a |
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| Name | BDBM312203 |
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| Synonyms: | US9604926, Compound CM-401 | US9724435, Compound CM-401 |
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| Type | Small organic molecule |
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| Emp. Form. | C24H25FN2O3 |
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| Mol. Mass. | 408.4653 |
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| SMILES | CC(=O)c1ccc2n(CCCCN3CCC(=CC3)c3ccc(F)cc3)c(=O)oc2c1 |c:15| |
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| Structure | 
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