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TargetMitogen-activated protein kinase 14
LigandBDBM13354
Substrate/Competitormyelin basic protein
Meas. Tech.p38alpha Kinase Enzyme Assay
pH7.4±n/a
Temperature295.15±n/a K
IC50 196±n/a nM
Citation Gill, ALFrederickson, MCleasby, AWoodhead, SJCarr, MGWoodhead, AJWalker, MTCongreve, MSDevine, LATisi, DO'Reilly, MSeavers, LCDavis, DJCurry, JAnthony, RPadova, AMurray, CWCarr, RAJhoti, H Identification of novel p38alpha MAP kinase inhibitors using fragment-based lead generation. J Med Chem48:414-26 (2005) [PubMed]  Article
More Info.:Get all data from this article,  Inhibition_Run data,   Solution Info,  Assay Method
 
Mitogen-activated protein kinase 14
Name:Mitogen-activated protein kinase 14
Synonyms:CSAID-binding protein | CSBP | CSBP1 | CSBP2 | CSPB1 | Cytokine suppressive anti-inflammatory drug-binding protein | MAP kinase 14 | MAP kinase MXI2 | MAP kinase p38 alpha | MAPK 14 | MAPK14 | MAX-interacting protein 2 | MK14_HUMAN | MXI2 | Mitogen-activated protein kinase p38 alpha | SAPK2A | Stress-activated protein kinase 2a | p38 MAP kinase alpha/beta
Type:Serine/threonine-protein kinase
Mol. Mass.:41286.76
Organism:Homo sapiens (Human)
Description:Q16539
Residue:360
Sequence:
MSQERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQ
SIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQ
KLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMT
GYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVG
TPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAA
QALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLDQEEMES
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BDBM13354
myelin basic protein
Name:myelin basic protein
Synonyms:myelin A1 protein
Type:Other Protein Type
Mol. Mass.:4541.90
Organism:Oryctolagus cuniculus (rabbit)
Description:n/a
Residue:42
Sequence:
fgsdrgapkr gsgkdhaart thygslpqks ghrpqdenpv vh
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