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TargetcAMP-dependent protein kinase catalytic subunit alpha [L49I]
LigandBDBM14029
Substrate/CompetitorKemptide
Meas. Tech.Kinase Activity Assay
pH6.8±n/a
Temperature298.15±n/a K
IC50 28000±0 nM
Km10000±n/a nM
Citation Bonn, SHerrero, SBreitenlechner, CBErlbruch, ALehmann, WEngh, RAGassel, MBossemeyer, D Structural analysis of protein kinase A mutants with Rho-kinase inhibitor specificity. J Biol Chem281:24818-30 (2006) [PubMed]  Article
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
cAMP-dependent protein kinase catalytic subunit alpha [L49I]
Name:cAMP-dependent protein kinase catalytic subunit alpha [L49I]
Synonyms:KAPCA_BOVIN | PKA C-alpha | PRKACA | cAMP-Dependent Protein Kinase (PKA) Mutant (L49I) | cAMP-Dependent Protein Kinase (PKA) Mutant PKAR1 (1) | cAMP-dependent protein kinase, alpha-catalytic subunit
Type:Enzyme Catalytic Subunit
Mol. Mass.:40627.77
Organism:Bos taurus (bovine)
Description:P00517[L49I]
Residue:351
Sequence:
MGNAAAAKKGSEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTIGTGSFGRVML
VKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMV
MEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGY
IQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFF
ADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFAT
TDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF
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  Blast E-value cutoff:
BDBM14029
Kemptide
Name:Kemptide
Synonyms:Aurora Peptide Substrate
Type:Peptide
Mol. Mass.:773.92
Organism:n/a
Description:50 uM ATP as co-substrate.
Residue:7
Sequence:
LRRASLG