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TargetcAMP-dependent protein kinase catalytic subunit alpha [V123M,Q181K,T183A]
LigandBDBM2579
Substrate/CompetitorKemptide
Meas. Tech.Kinase Activity Assay
IC50<45±n/a nM
Citation Bonn, SHerrero, SBreitenlechner, CBErlbruch, ALehmann, WEngh, RAGassel, MBossemeyer, D Structural analysis of protein kinase A mutants with Rho-kinase inhibitor specificity. J Biol Chem281:24818-30 (2006) [PubMed]  Article
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
cAMP-dependent protein kinase catalytic subunit alpha [V123M,Q181K,T183A]
Name:cAMP-dependent protein kinase catalytic subunit alpha [V123M,Q181K,T183A]
Synonyms:KAPCA_BOVIN | PKA C-alpha | PRKACA | cAMP-Dependent Protein Kinase (PKA) Mutant (V123M/Q181K/T183A) | cAMP-Dependent Protein Kinase (PKA) Mutant PKAR3 (1) | cAMP-dependent protein kinase, alpha-catalytic subunit
Type:Enzyme Catalytic Unit
Mol. Mass.:40630.86
Organism:Bos taurus (bovine)
Description:P00517[V123M,Q181K,T183A]
Residue:351
Sequence:
MGNAAAAKKGSEQESVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVML
VKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMV
MEYMPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGY
IKVADFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFF
ADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFAT
TDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM2579
Kemptide
Name:Kemptide
Synonyms:Aurora Peptide Substrate
Type:Peptide
Mol. Mass.:773.92
Organism:n/a
Description:50 uM ATP as co-substrate.
Residue:7
Sequence:
LRRASLG