Reaction Details |
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Target | Mitogen-activated protein kinase 14 [G110D] |
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Ligand | BDBM15244 |
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Substrate/Competitor | biotinylated GST-ATF2 |
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Meas. Tech. | Enzyme Inhibition Scintillation Proximity Assay |
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pH | 7±n/a |
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Temperature | 303.15±n/a K |
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IC50 | 120±n/a nM |
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Km | 48000±4000 nM |
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Citation | Fitzgerald, CE; Patel, SB; Becker, JW; Cameron, PM; Zaller, D; Pikounis, VB; O'Keefe, SJ; Scapin, G Structural basis for p38alpha MAP kinase quinazolinone and pyridol-pyrimidine inhibitor specificity. Nat Struct Biol10:764-9 (2003) [PubMed] Article |
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More Info.: | Get all data from this article, Inhibition_Run data, Solution Info, Assay Method |
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Mitogen-activated protein kinase 14 [G110D] |
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Name: | Mitogen-activated protein kinase 14 [G110D] |
Synonyms: | Crk1 | Csbp1 | Csbp2 | MAP Kinase p38 alpha Mutant (G110D) | MK14_MOUSE | Mapk14 | Mitogen-activated protein kinase 14 | Mitogen-activated protein kinase p38 alpha |
Type: | Enzyme |
Mol. Mass.: | 41338.25 |
Organism: | Mus musculus (mouse) |
Description: | Mutant was site-directed generated from wild-type p38alpha. |
Residue: | 360 |
Sequence: | MSQERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGHRVAVKKLSRPFQ
SIIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMDADLNNIVKCQ
KLTDDHVQFLIYQILRGLKYIHSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMT
GYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRTLFPGTDHIDQLKLILRLVG
TPGAELLKKISSESARNYIQSLAQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAA
QALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLDQEEMES
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BDBM15244 |
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biotinylated GST-ATF2 |
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Name: | biotinylated GST-ATF2 |
Synonyms: | ATF-2-GST | ATF2 | Activating transcription factor 2 | Activating transcription factor 2-GST fusion | GST-ATF2 | biotinylated ATF2 substrate | biotinylated activating transcription factor 2 |
Type: | Other Protein Type |
Mol. Mass.: | 12237.77 |
Organism: | Homo sapiens (Human) |
Description: | n/a |
Residue: | 109 |
Sequence: | MSDDKPFLCTAPGCGQRFTNEDHLAVHKHKHEMTLKFGPARNDSVIVADQTPTPTRFLKN
CEEVGLFNELASPFENEFKKASEDDIKKMPLDLSPLATPIIRSKIEEPS
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